SCHEMBL6409574

SCHEMBL6409574

O=C(NC1CCCC1)OC1=NOC2(CCN(C(=O)c3cccnc3Oc3ccccc3)CC2)C1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
RAB9A P51151 1/20 0.40
POLB P06746 1/20 0.40
CNR2 P34972 2/20 0.39
CNR1 P21554 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
EPHX2 P34913 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2401286 0.87 CNR2 (0.44) ALDH1A1POLBCNR2CNR1TDP1
SCHEMBL6416605 0.86 POLB (0.43) ALDH1A1RAB9APOLBTDP1EPHX2
SCHEMBL6409707 0.85 MAPK8 (0.51) ALDH1A1
SCHEMBL15309149 0.79 TDP1 (0.44) ALDH1A1POLBTDP1
SCHEMBL2403591 0.74 MAPK8 (0.57) ALDH1A1
SCHEMBL2400992 0.73 TDP1 (0.46) ALDH1A1POLBTDP1
SCHEMBL6412218 0.73 ALDH1A1 (0.40) ALDH1A1RAB9APOLB
SCHEMBL6410889 0.73 MAPT (0.39) ALDH1A1POLBTDP1EPHX2
SCHEMBL2583086 0.71 CYP2C19 (0.44) ALDH1A1RAB9APOLBCNR2CNR1
SCHEMBL6411430 0.69 RAB9A (0.47) ALDH1A1RAB9APOLBTDP1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401841-B1 SUBSTITUTED 1-OXA-2,8-DIAZA-SPIRO 4,5]DEC-2-ENE DERIVATIVES AS MEDICAMENTS FOR THE TREATMENT OF PAIN GRUENENTHAL GMBH (DE) 2005-08-24 EP claimed
EP-1521828-A2 PRODUCTION OF POLYKETIDES Biotica Technology Limited (GB) 2005-04-13 EP claimed
WO-2004007709-A2 PRODUCTION OF POLYKETIDES BIOTICA TECHNOLOGY LIMITED (GB) 2004-01-22 WO claimed
EP-1401841-B1 SUBSTITUTED 1-OXA-2,8-DIAZA-SPIRO 4,5]DEC-2-ENE DERIVATIVES AS MEDICAMENTS FOR THE TREATMENT OF PAIN GRUENENTHAL GMBH (DE) 2005-08-24 EP disclosed