SCHEMBL6411896

SCHEMBL6411896

O=C(NC(CCN1CCC2(CC1)CCN(Cc1ccc(Br)cc1)C2=O)c1ccccc1)c1ccncc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 6/20 0.54
ROCK2 O75116 4/20 0.54
UTS2R Q9UKP6 4/20 0.46
GSK3B P49841 4/20 0.42
CLK4 Q9HAZ1 4/20 0.42
GSK3A P49840 3/20 0.42
PRKACA P17612 2/20 0.42
PRKX P51817 2/20 0.42
PRKCQ Q04759 2/20 0.42
CDK8 P49336 1/20 0.42
CCR5 P51681 4/20 0.41
RPS6KA5 O75582 3/20 0.39
AKT1 P31749 3/20 0.39
NEK4 P51957 3/20 0.39
PRKCD Q05655 3/20 0.39
PRKG2 Q13237 3/20 0.39
PRKG1 Q13976 3/20 0.39
PKN2 Q16513 3/20 0.39
MAPK13 O15264 2/20 0.39
MAP4K4 O95819 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6414705 0.99 ROCK1 (0.54) ROCK1ROCK2UTS2RGSK3BCLK4
SCHEMBL6408477 0.94 UTS2R (0.52) ROCK1ROCK2UTS2RCCR5HDAC1
Hydrochloric Acid SCHEMBL6412861 0.93 UTS2R (0.51) ROCK1ROCK2UTS2RCCR5HDAC1
SCHEMBL6418852 0.91 ROCK2 (0.46) ROCK1ROCK2UTS2RCCR5MAPK1
SCHEMBL6413738 0.91 UTS2R (0.55) ROCK1ROCK2UTS2RCCR5HDAC1
Hydrochloric Acid SCHEMBL6416620 0.90 ROCK2 (0.45) ROCK1ROCK2UTS2RCCR5MAPK1
Hydrochloric Acid SCHEMBL6409140 0.90 UTS2R (0.55) ROCK1ROCK2UTS2RCCR5HDAC1
SCHEMBL6409097 0.90 ROCK2 (0.55) ROCK1ROCK2UTS2RGSK3BCLK4
Hydrochloric Acid SCHEMBL6409114 0.89 ROCK2 (0.54) ROCK1ROCK2UTS2RGSK3BCLK4
SCHEMBL6410740 0.89 ROCK1 (0.51) ROCK1ROCK2UTS2RGSK3BCLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050075326-A1 Spiro compounds and methods for the modulation of chemokine receptor activity VIROCHEM PHARMA INC (CA) 2005-04-07 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050075326-A1 Spiro compounds and methods for the modulation of chemokine receptor activity CXCR1, CXCR4, CXCR2 ROCK1 1002/4885ROCK2 1735/4885UTS2R 126/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.