SCHEMBL6413337

SCHEMBL6413337

COc1ccc2c(n1)C(=O)c1ncc(OC)c(C)c1C2=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 3/20 0.36
G6PD P11413 2/20 0.36
DNMT1 P26358 2/20 0.36
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
WEE1 P30291 1/20 0.34
MAPT P10636 6/20 0.34
KMT2A Q03164 5/20 0.34
MEN1 O00255 4/20 0.34
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 3/20 0.34
TDP1 Q9NUW8 2/20 0.34
USP2 O75604 1/20 0.34
DUSP3 P51452 1/20 0.34
MAOA P21397 1/20 0.33
RAB9A P51151 4/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
NPC1 O15118 3/20 0.33
USP8 P40818 2/20 0.33
USP7 Q93009 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6410254 0.95 NSD2 (0.36) NSD2G6PDDNMT1ADORA2AADORA1
SCHEMBL6407781 0.80 S100A4 (0.50) NSD2MAPTKMT2AMEN1ALDH1A1
SCHEMBL6408454 0.78 NSD2 (0.40) NSD2G6PDDNMT1ADORA2AADORA1
SCHEMBL6410278 0.74 MAPT (0.36) G6PDMAPTKMT2AMEN1ALDH1A1
SCHEMBL6415723 0.74 S100A4 (0.50) NSD2KMT2AMEN1TDP1BLM
SCHEMBL6408521 0.73 LMNA (0.42) MAPTKMT2AKDM4ETDP1MAOA
SCHEMBL6414247 0.73 MAPT (0.37) G6PDMAPTKMT2AMEN1ALDH1A1
SCHEMBL6413377 0.72 NSD2 (0.40) NSD2G6PDDNMT1MAPTKMT2A
SCHEMBL6410373 0.71 MAPT (0.36) G6PDMAPTKMT2AALDH1A1KDM4E
SCHEMBL6407769 0.70 LMNA (0.44) MAPTKMT2AKDM4ETDP1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1202993-B1 PHENANTHROLINE-7-ONE DERIVATIVES AND THEIR THERAPEUTIC USES LAFON LABOR (FR) 2005-10-19 EP disclosed
US-6809096-B1 SUCH AS 11-METHOXY-7H-PYRIDO(4,3,2-DE)(1,7)PHENANTHROLINE-7-ONE; ANTITUMOR AGENTS LABORATOIRE L. LAFON (FR) 2004-10-26 US disclosed
EP-1202993-A2 PHENANTHROLINE-7-ONE DERIVATIVES AND THEIR THERAPEUTIC USES LABORATOIRE L. LAFON (FR) 2002-05-08 EP disclosed
WO-2001012632-A2 PHENANTHROLINE-7-ONE DERIVATIVES AND THEIR THERAPEUTIC USES LABORATOIRE L. LAFON (FR) 2001-02-22 WO disclosed