SCHEMBL6421885

SCHEMBL6421885

CC(C)n1c2c(c3ccccc31)CCN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
CHRM2 P08172 1/20 0.45
CHRM4 P08173 1/20 0.45
CHRM1 P11229 1/20 0.45
CHRM3 P20309 1/20 0.45
ESR2 Q92731 1/20 0.43
NR1H2 P55055 2/20 0.42
MAPK1 P28482 1/20 0.42
HTR6 P50406 1/20 0.41
F12 P00748 1/20 0.41
ADORA1 P30542 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
KRAS P01116 1/20 0.40
DDB1 Q16531 1/20 0.40
CRBN Q96SW2 1/20 0.40
PDK4 Q16654 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
PARP1 P09874 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28606605 0.91 HDAC1 (0.57) HDAC1HDAC6CHRM2CHRM4CHRM1
SCHEMBL969755 0.85 HDAC6 (0.52) HDAC1HDAC6CHRM2CHRM4CHRM1
SCHEMBL6422033 0.83 CHRM2 (0.51) HDAC1HDAC6CHRM2CHRM4CHRM1
SCHEMBL6422069 0.82 HDAC1 (0.51) HDAC1HDAC6CHRM2CHRM4CHRM1
SCHEMBL968966 0.82 HDAC1 (0.50) HDAC1HDAC6CHRM2CHRM4CHRM1
SCHEMBL6421557 0.82 HDAC1 (0.52) HDAC1HDAC6CHRM2CHRM4CHRM1
SCHEMBL6423913 0.82 HDAC1 (0.50) HDAC1HDAC6CHRM2CHRM4CHRM1
SCHEMBL6421798 0.80 HDAC1 (0.55) HDAC1HDAC6CHRM2CHRM4CHRM1
SCHEMBL6421094 0.80 PTGDR2 (0.59) HDAC1HDAC6CHRM2CHRM4CHRM1
SCHEMBL6420928 0.80 HDAC1 (0.51) HDAC1HDAC6CHRM2CHRM4CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1057814-B1 TETRAHYDROBENZINDOLE DERIVATIVES MEIJI SEIKA KAISHA (JP) 2005-03-09 EP disclosed
US-6498251-B1 Tetrahydrobenzindole derivatives MEIJI SEIKA KAISHA, LTD. (JP) 2002-12-24 US disclosed
EP-1057814-A1 TETRAHYDROBENZINDOLE DERIVATIVES Meiji Seika Kaisha, Ltd. (JP) 2000-12-06 EP disclosed