SCHEMBL6422780

SCHEMBL6422780

C=CCn1c2c(c3ccccc31)CCNC2

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.52
HDAC6 Q9UBN7 2/20 0.52
HTR6 P50406 5/20 0.49
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
KDM4E B2RXH2 1/20 0.47
ALOX15 P16050 1/20 0.47
MAPK1 P28482 1/20 0.47
HSD17B10 Q99714 1/20 0.47
GAA P10253 1/20 0.42
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
HTR3A P46098 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
HTR7 P34969 1/20 0.39
KRAS P01116 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6038551 0.90 HTR2C (0.56) HDAC1HDAC6HTR6HTR2AHTR2C
SCHEMBL4300297 0.82 HDAC1 (0.53) HDAC1HDAC6HTR6HTR2AHTR2C
SCHEMBL9615137 0.81 HTR2A (0.55) HDAC1HDAC6HTR6HTR2AHTR2C
Hydrochloric Acid SCHEMBL9696491 0.80 KDM4E (0.56) HDAC1HDAC6HTR6HTR2AHTR2C
SCHEMBL9903966 0.80 CA1 (0.65) HDAC1HDAC6HTR6HTR2AHTR2C
SCHEMBL6422248 0.79 HDAC1 (0.69) HDAC1HDAC6HTR6HTR2AHTR2C
SCHEMBL6422112 0.78 HTR2C (0.55) HDAC1HDAC6HTR6HTR2AHTR2C
Hydrochloric Acid SCHEMBL9615118 0.78 HDAC1 (0.67) HDAC1HDAC6HTR6HTR2AHTR2C
SCHEMBL12369406 0.76 HDAC1 (0.53) HDAC1HDAC6HTR6HTR2AHTR2C
SCHEMBL9615110 0.76 NPC1 (0.54) HDAC1HDAC6HTR6HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1057814-B1 TETRAHYDROBENZINDOLE DERIVATIVES MEIJI SEIKA KAISHA (JP) 2005-03-09 EP disclosed
US-6498251-B1 Tetrahydrobenzindole derivatives MEIJI SEIKA KAISHA, LTD. (JP) 2002-12-24 US disclosed
EP-1057814-A1 TETRAHYDROBENZINDOLE DERIVATIVES Meiji Seika Kaisha, Ltd. (JP) 2000-12-06 EP disclosed