SCHEMBL6423547

SCHEMBL6423547

CN1CCN(C(=O)[C@H](CNC(=O)OC(C)(C)C)NC(=O)O)CC1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.38
SIGMAR1 Q99720 3/20 0.38
CYP2C19 P33261 1/20 0.37
CTSS P25774 2/20 0.37
CTSK P43235 2/20 0.37
CTSL P07711 1/20 0.37
CTSB P07858 1/20 0.37
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
ALDH1A1 P00352 2/20 0.37
ITGB3 P05106 2/20 0.37
ITGA2B P08514 2/20 0.37
GAA P10253 1/20 0.37
HRH2 P25021 2/20 0.36
HRH1 P35367 2/20 0.36
TGM2 P21980 1/20 0.36
MAPK1 P28482 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14850693 0.92 TSHR (0.41) TSHRCTSSCTSKCTSLCTSB
SCHEMBL16435346 0.86 CTSS (0.45) TSHRCTSSCTSKCTSLCTSB
SCHEMBL3500871 0.86 USP2 (0.44) TSHRCYP2C19CTSSCTSKCTSL
SCHEMBL3492474 0.86 USP2 (0.44) TSHRCYP2C19CTSSCTSKCTSL
SCHEMBL14850788 0.83 ITGB3 (0.45) TSHRCTSSCTSKCTSLCTSB
SCHEMBL14497033 0.81 SYK (0.60) CTSKALDH1A1ITGB3ITGA2BTGM2
SCHEMBL14850864 0.81 ITGB3 (0.46) TSHRCTSSCTSKCTSLCTSB
SCHEMBL14850855 0.80 ITGB3 (0.47) TSHRCTSSCTSKCTSLCTSB
SCHEMBL14850692 0.80 ITGB3 (0.47) TSHRCTSSCTSKCTSLCTSB
SCHEMBL16435373 0.80 HRH2 (0.47) TSHRSIGMAR1CTSSCTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1577302-A1 NOVEL ETHYLENEDIAMINE DERIVATIVES DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2005-09-21 EP disclosed