SCHEMBL6423607

SCHEMBL6423607

COc1ccc(C=C(C(=O)O)c2ccc(O)cc2)cc1OC.COc1ccc(CC(C(=O)O)c2ccc(O)cc2)cc1OC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.53
HTT P42858 1/20 0.53
AKR1C3 P42330 1/20 0.51
LDHA P00338 1/20 0.47
PTPN7 P35236 1/20 0.43
PTPN12 Q05209 1/20 0.43
PTPN22 Q9Y2R2 1/20 0.43
AKR1C2 P52895 1/20 0.43
MME P08473 1/20 0.43
MMP1 P03956 7/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
POLB P06746 1/20 0.43
MMP2 P08253 2/20 0.42
MMP3 P08254 2/20 0.42
MMP9 P14780 2/20 0.42
MMP12 P39900 2/20 0.42
MMP13 P45452 2/20 0.42
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6423606 1.00 KDM4E (0.53) KDM4EHTTAKR1C3LDHAPTPN7
SCHEMBL6423609 0.85 ESR1 (0.46) KDM4EHTTAKR1C3LDHAPDE4A
SCHEMBL4658405 0.85 LDHA (0.64) HTTLDHAMMEMMP1KMT2A
SCHEMBL4659113 0.84 AKR1C3 (0.68) KDM4EHTTAKR1C3AKR1C2KMT2A
SCHEMBL4659114 0.84 AKR1C3 (0.68) KDM4EHTTAKR1C3AKR1C2KMT2A
SCHEMBL5314275 0.75 KDM4E (0.80) KDM4EHTTAKR1C3AKR1C2KMT2A
SCHEMBL5314277 0.75 KDM4E (0.80) KDM4EHTTAKR1C3AKR1C2KMT2A
SCHEMBL28659073 0.74 AKR1C3 (0.68) KDM4EHTTAKR1C3AKR1C2KMT2A
SCHEMBL3047079 0.74 AKR1C3 (0.72) KDM4EHTTAKR1C3AKR1C2KMT2A
SCHEMBL30159708 0.74 AKR1C3 (0.68) KDM4EHTTAKR1C3AKR1C2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1251738-A4 NOVEL DIPHENYLETHYLENE COMPOUNDS CALYX THERAPEUTICS INC (US) 2005-08-10 EP disclosed
EP-1251738-A1 NOVEL DIPHENYLETHYLENE COMPOUNDS Calyx Therapeutics, Inc. (US) 2002-10-30 EP disclosed
WO-2001056382-A1 NOVEL DIPHENYLETHYLENE COMPOUNDS CALYX THERAPEUTICS, INC. (US) 2001-08-09 WO disclosed