SCHEMBL6423609

SCHEMBL6423609

COc1ccc(C=C(C(=O)OC(=O)C(Cc2ccc(OC)c(OC)c2)c2ccc(O)cc2)c2ccc(O)cc2)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.46
ESR2 Q92731 1/20 0.46
HTT P42858 2/20 0.42
KDM4E B2RXH2 1/20 0.42
PTGS1 P23219 2/20 0.42
ALDH1A1 P00352 4/20 0.41
PKM P14618 1/20 0.41
LDHA P00338 1/20 0.41
EGFR P00533 1/20 0.41
AKR1C3 P42330 1/20 0.41
LMNA P02545 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
SLC22A1 O15245 1/20 0.41
ADRB2 P07550 1/20 0.41
CHRM2 P08172 1/20 0.41
ADRB1 P08588 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6423606 0.85 KDM4E (0.53) ESR1ESR2HTTKDM4EALDH1A1
SCHEMBL6423607 0.85 KDM4E (0.53) ESR1ESR2HTTKDM4EALDH1A1
SCHEMBL4658405 0.75 LDHA (0.64) ESR1ESR2HTTALDH1A1LDHA
SCHEMBL4659114 0.73 AKR1C3 (0.68) HTTKDM4EPTGS1ALDH1A1AKR1C3
SCHEMBL4659113 0.73 AKR1C3 (0.68) HTTKDM4EPTGS1ALDH1A1AKR1C3
SCHEMBL27948969 0.70 PDE4A (0.53) HTTKDM4EPTGS1ALDH1A1AKR1C3
SCHEMBL28673604 0.70 PDE4A (0.53) HTTKDM4EPTGS1ALDH1A1AKR1C3
SCHEMBL3051689 0.68 NQO2 (0.63) HTTKDM4EALDH1A1AKR1C3PDE4A
SCHEMBL28673508 0.68 AKR1C3 (0.53) HTTKDM4EALDH1A1PKMAKR1C3
SCHEMBL3049032 0.68 NQO2 (0.63) HTTKDM4EALDH1A1AKR1C3PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1251738-A4 NOVEL DIPHENYLETHYLENE COMPOUNDS CALYX THERAPEUTICS INC (US) 2005-08-10 EP disclosed
EP-1251738-A1 NOVEL DIPHENYLETHYLENE COMPOUNDS Calyx Therapeutics, Inc. (US) 2002-10-30 EP disclosed
WO-2001056382-A1 NOVEL DIPHENYLETHYLENE COMPOUNDS CALYX THERAPEUTICS, INC. (US) 2001-08-09 WO disclosed