SCHEMBL6424933

SCHEMBL6424933

O=C(O)c1cc2c(s1)CNCCC2

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.65
DAO P14920 1/20 0.65
PNMT P11086 2/20 0.49
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C19 P33261 2/20 0.42
POLB P06746 2/20 0.42
PKM P14618 1/20 0.42
CYP3A4 P08684 1/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 4/20 0.41
TP53 P04637 1/20 0.41
MAPK1 P28482 1/20 0.41
ITGB3 P05106 2/20 0.41
ITGA2B P08514 2/20 0.41
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP2C9 P11712 1/20 0.39
KDM4E B2RXH2 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1173969 0.90 ALDH1A1 (0.59) ALDH1A1DAOPNMTHPGDITGB3
SCHEMBL6421249 0.87 ALDH1A1 (0.65) ALDH1A1DAOPNMTMEN1KMT2A
SCHEMBL2761783 0.85 KDM4E (0.54) ALDH1A1DAOPNMTMEN1KMT2A
SCHEMBL977949 0.80 PNMT (0.73) ALDH1A1DAOPNMTITGB3ITGA2B
Hydrochloric Acid SCHEMBL19712091 0.80 ALDH1A1 (0.53) ALDH1A1DAOPNMTMEN1KMT2A
SCHEMBL2954334 0.79 DAO (1.00) ALDH1A1DAOMEN1KMT2ACYP1A2
SCHEMBL1068704 0.79 ALDH1A1 (1.00) ALDH1A1DAOMEN1KMT2ACYP1A2
Hydrochloric Acid SCHEMBL3441470 0.79 PNMT (0.71) ALDH1A1DAOPNMTITGB3ITGA2B
SCHEMBL11174836 0.78 ALDH1A1 (0.66) ALDH1A1DAOPNMTMEN1KMT2A
SCHEMBL3743711 0.78 ALDH1A1 (0.96) ALDH1A1DAOMEN1KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1057814-B1 TETRAHYDROBENZINDOLE DERIVATIVES MEIJI SEIKA KAISHA (JP) 2005-03-09 EP disclosed
US-6498251-B1 Tetrahydrobenzindole derivatives MEIJI SEIKA KAISHA, LTD. (JP) 2002-12-24 US disclosed
US-6407112-B1 2A,3,4,5-TETRAHYDRO-1H-BENZ(CD)INDOL-2-ONE DERIVATIVES; 5-HYDROXYTRYPTAMINE AGONISTS; SLEEP, CIRCADIAN RHYTHYM, BIPOLAR, AND PSYCHOLOGICAL DISORDER TREATMENT MEIJI SEIKA KAISHA, LTD. (JP) 2002-06-18 US disclosed
EP-1081136-A1 OPTICALLY ACTIVE TETRAHYDROBENZINDOLE DERIVATIVES Meiji Seika Kaisha, Ltd. (JP) 2001-03-07 EP disclosed
EP-1057814-A1 TETRAHYDROBENZINDOLE DERIVATIVES Meiji Seika Kaisha, Ltd. (JP) 2000-12-06 EP disclosed