SCHEMBL6427643

SCHEMBL6427643

O=C(OC(=O)c1cc([N+](=O)[O-])cc([N+](=O)[O-])c1)c1ccccc1

nearest known ligand 0.69

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 7/20 0.69
CES2 O00748 3/20 0.56
CES1 P23141 2/20 0.56
PTGES O14684 1/20 0.55
TP53 P04637 1/20 0.54
CYP3A4 P08684 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
KDM4E B2RXH2 1/20 0.50
GAA P10253 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
PTPN2 P17706 1/20 0.49
PTPN1 P18031 1/20 0.49
PTPN6 P29350 1/20 0.49
PTPN11 Q06124 1/20 0.49
ATM Q13315 1/20 0.49
ALDH1A1 P00352 2/20 0.49
TSHR P16473 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6427641 0.89 CYP3A4 (0.61) ALOX5CES2CES1PTGESTP53
SCHEMBL4721016 0.88 TP53 (0.67) ALOX5CES2CES1TP53SMN1; SMN2
SCHEMBL254774 0.86 CES1 (0.70) ALOX5CES2CES1TDP1ALDH1A1
Methane SCHEMBL28800504 0.84 CES1 (0.68) ALOX5CES2CES1TDP1ALDH1A1
SCHEMBL11842226 0.83 ALOX5 (0.56) ALOX5CES2CES1PTGESTP53
SCHEMBL14893088 0.83 ALOX5 (0.49) ALOX5CES2CES1TP53SMN1; SMN2
SCHEMBL4721013 0.82 CES2 (0.70) ALOX5CES2CES1TP53CYP3A4
SCHEMBL6911469 0.82 CES2 (0.75) ALOX5CES2CES1TP53CYP3A4
SCHEMBL27935077 0.81 ALOX5 (1.00) ALOX5CES2CES1PTGESKDM4E
SCHEMBL27971368 0.81 ALOX5 (0.77) ALOX5CES2CES1PTGESTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1387822-B1 2-[4-(2,2,-DIHALOCYCLOPROPYL)PHENOXY]-ALKANOIC ACIDS AND ESTERS THEREOF PRODUCTION PROCESS LABORATORIO CHIMICO INT SPA (IT) 2005-06-15 EP claimed
EP-1387822-A1 2-[4-(2,2,-DIHALOCYCLOPROPYL)PHENOXY]-ALKANOIC ACIDS AND ESTERS THEREOF PRODUCTION PROCESS LABORATORIO CHIMICO INTERNAZIONALE S.p.A. (IT) 2004-02-11 EP claimed
WO-2002090307-A1 2-[4-(2, 2-DIHALOCYCLOPROPYL)PHENOXY]-ALKANOIC ACIDS AND ESTERS THEREOF PRODUCTION PROCESS LABORATORIO CHIMICO INTERNAZIONALE S.P.A. (IT) 2002-11-14 WO claimed
CN-104059068-B Beta-amino-carbonyl compound, preparation method, its pharmaceutical composition and application thereof 中国科学院上海药物研究所 2017-02-08 CN disclosed
CN-104059068-A Beta-amino-carbonyl compound, preparation method, its pharmaceutical composition and application thereof SHANGHAI INST MATERIA MEDICA 2014-09-24 CN disclosed
EP-1387822-B1 2-[4-(2,2,-DIHALOCYCLOPROPYL)PHENOXY]-ALKANOIC ACIDS AND ESTERS THEREOF PRODUCTION PROCESS LABORATORIO CHIMICO INT SPA (IT) 2005-06-15 EP disclosed