SCHEMBL6428631

SCHEMBL6428631

CCOC(=O)c1ccc(/C=C(/c2ccc3c(c2)C(C)(C)CCC3(C)C)[Si](C)(C)C)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 15/20 0.53
RARB P10826 14/20 0.53
RARG P13631 13/20 0.53
RXRA P19793 7/20 0.50
CYP3A4 P08684 4/20 0.50
CYP26A1 O43174 4/20 0.50
KDM4E B2RXH2 1/20 0.50
NPC1 O15118 1/20 0.50
GMNN O75496 1/20 0.50
USP2 O75604 1/20 0.50
ALDH1A1 P00352 1/20 0.50
LMNA P02545 1/20 0.50
TP53 P04637 1/20 0.50
CYP1A2 P05177 1/20 0.50
POLB P06746 1/20 0.50
CYP2D6 P10635 1/20 0.50
NFKB1 P19838 1/20 0.50
CYP2C19 P33261 1/20 0.50
THPO P40225 1/20 0.50
MTOR P42345 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28749819 1.00 RARA (0.53) RARARARBRARGRXRACYP3A4
SCHEMBL27582113 0.88 RXRA (0.53) RARARARBRARGRXRACYP26A1
SCHEMBL6429289 0.88 RXRA (0.53) RARARARBRARGRXRACYP26A1
Arotinoid SCHEMBL2890175 0.85 RARG (0.70) RARARARBRARGRXRACYP3A4
Arotinoid SCHEMBL29430179 0.85 RARG (0.70) RARARARBRARGRXRACYP3A4
Arotinoid SCHEMBL2890176 0.85 RARG (0.70) RARARARBRARGRXRACYP3A4
SCHEMBL11256000 0.84 RARB (0.52) RARARARBRARGRXRACYP3A4
SCHEMBL11256004 0.84 RARB (0.52) RARARARBRARGRXRACYP3A4
SCHEMBL6258868 0.83 RARB (0.70) RARARARBRARGRXRACYP3A4
SCHEMBL6258870 0.83 RARB (0.70) RARARARBRARGRXRACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6906057-B1 Methods for modulating FXR receptor activity ALLERGAN, INC. (US) 2005-06-14 US disclosed