SCHEMBL6428878

SCHEMBL6428878

COc1ccc(CNC(=O)c2cc3c(=O)n(C(C)c4ccc(C(=O)O)c(C)c4)c(=O)[nH]c3cn2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 4/20 0.49
SLC22A8 Q8TCC7 1/20 0.49
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ALDH1A1 P00352 4/20 0.43
HPGD P15428 3/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
POLB P06746 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C19 P33261 1/20 0.43
ATM Q13315 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
KDM4E B2RXH2 3/20 0.42
PKM P14618 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
MAPT P10636 1/20 0.41
EGLN3 Q9H6Z9 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6238392 0.91 MMP13 (0.57) MMP13SLC22A8MEN1KMT2AALDH1A1
SCHEMBL6235396 0.88 MEN1 (0.52) MMP13MEN1KMT2AALDH1A1CYP3A4
SCHEMBL6238386 0.88 MMP13 (0.49) MMP13SLC22A8MEN1KMT2AALDH1A1
SCHEMBL6235291 0.82 MMP13 (0.58) MMP13SLC22A8
SCHEMBL7104022 0.82 MMP13 (0.45) MMP13SLC22A8MEN1KMT2AALDH1A1
SCHEMBL6727454 0.81 MEN1 (0.50) MMP13MEN1KMT2AALDH1A1CYP3A4
SCHEMBL6236712 0.81 MEN1 (0.52) MMP13MEN1KMT2AALDH1A1CYP3A4
SCHEMBL6238482 0.81 MEN1 (0.51) MMP13MEN1KMT2AALDH1A1CYP3A4
SCHEMBL6232533 0.81 MEN1 (0.53) MMP13MEN1KMT2AALDH1A1CYP3A4
SCHEMBL7624017 0.80 MEN1 (0.51) MMP13MEN1KMT2AALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530467-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB Warner-Lambert Company LLC (US) 2005-05-18 EP disclosed
WO-2004006912-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed