SCHEMBL6429533

SCHEMBL6429533

CC(C)(C)Oc1ccc(C[C@H](NC(=O)[C@@H]2CCCN2S(=O)(=O)Cc2ccccc2)C(=O)O)cc1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 6/20 0.52
ITGA5 P08648 2/20 0.52
FKBP1A P62942 6/20 0.50
ITGA4 P13612 4/20 0.49
ITGB7 P26010 1/20 0.49
CCR4 P51679 1/20 0.48
CMA1 P23946 2/20 0.47
MMP8 P22894 1/20 0.46
MMP12 P39900 1/20 0.46
MMP13 P45452 1/20 0.46
ITGAV P06756 1/20 0.45
ITGA2 P17301 1/20 0.45
YAP1 P46937 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7070239 0.89 FKBP1A (0.61) ITGB1ITGA5FKBP1AITGA4ITGB7
SCHEMBL6429378 0.88 ITGB1 (0.67) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL6637622 0.84 ITGB1 (0.57) ITGB1ITGA5FKBP1AITGA4ITGB7
SCHEMBL6368426 0.83 ITGB1 (0.58) ITGB1ITGA5ITGA4ITGB7MMP13
SCHEMBL6431309 0.83 ITGB1 (0.58) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL7707493 0.83 ITGB1 (0.60) ITGB1ITGA5FKBP1AITGA4ITGB7
SCHEMBL5690343 0.82 ITGB1 (0.53) ITGB1ITGA5ITGA4CMA1ITGAV
SCHEMBL6634618 0.82 ITGB1 (0.50) ITGB1ITGA5FKBP1AITGA4ITGB7
SCHEMBL6367886 0.82 ITGB1 (0.55) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL6367527 0.82 ITGB1 (0.71) ITGB1ITGA5ITGA4ITGB7ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP claimed
JP-2002512625-A 2002-04-23 JP claimed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP claimed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO claimed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed