SCHEMBL5690343

SCHEMBL5690343

CC(C)(C)OC(=O)N1CCC(C(=O)Nc2ccc(C[C@H](NC(=O)[C@@H]3CCCN3S(=O)(=O)Cc3ccccc3)C(=O)O)cc2)CC1

nearest known ligand 0.66

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 4/20 0.53
ITGA5 P08648 2/20 0.53
MAPK1 P28482 1/20 0.53
STS P08842 1/20 0.53
YAP1 P46937 2/20 0.50
PTPN2 P17706 1/20 0.49
PTPN1 P18031 1/20 0.49
PTPN6 P29350 1/20 0.49
PABPC1 P11940 1/20 0.47
ABL1 P00519 1/20 0.47
RIN1 Q13671 1/20 0.47
KMT2A Q03164 2/20 0.46
ITGAV P06756 1/20 0.46
CMA1 P23946 2/20 0.45
ITGA4 P13612 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5691845 0.93 MAPT (0.50) ITGB1ITGA5MAPK1STSYAP1
SCHEMBL5690885 0.86 ITGB1 (0.58) ITGB1ITGA5MAPK1PTPN2PTPN1
SCHEMBL5690351 0.85 ITGB1 (0.58) ITGB1ITGA5ITGAVITGA4MAPT
SCHEMBL6429533 0.82 ITGB1 (0.52) ITGB1ITGA5YAP1ITGAVCMA1
SCHEMBL7070239 0.82 FKBP1A (0.61) ITGB1ITGA5ITGA4
SCHEMBL6165579 0.81 MAPK1 (0.75) MAPK1STSYAP1KMT2A
SCHEMBL6165580 0.81 MAPK1 (0.75) MAPK1STSYAP1KMT2A
SCHEMBL5690979 0.80 ALDH1A1 (0.53) ITGB1ITGA5MAPK1YAP1ITGAV
SCHEMBL5690719 0.80 ITGB1 (0.57) ITGB1ITGA5MAPK1ITGAVITGA4
SCHEMBL5691083 0.80 ITGB1 (0.48) ITGB1ITGA5ITGAVCMA1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001974-B1 4-AMINO-PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARM INC (US) 2006-05-24 EP claimed