SCHEMBL6433087

SCHEMBL6433087

N/N=C(\c1ccc(C(=O)O)cc1)c1nc2nonc2nc1NCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
POLB P06746 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CTDSP1 Q9GZU7 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NPSR1 Q6W5P4 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
GAA P10253 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
VCP P55072 1/20 0.39
LDHA P00338 1/20 0.39
LDHB P07195 1/20 0.39
CSNK2A2 P19784 2/20 0.39
CSNK2A1 P68400 2/20 0.39
CSNK2B P67870 1/20 0.39
ACHE P22303 2/20 0.38
PLAU P00749 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6433104 1.00 ALDH1A1 (0.41) ALDH1A1POLBHPGDHSD17B10CTDSP1
SCHEMBL6416068 0.91 LDHA (0.46) NPSR1CYP1A2CYP3A4GAACYP2C9
SCHEMBL6416054 0.91 LDHA (0.46) NPSR1CYP1A2CYP3A4GAACYP2C9
SCHEMBL6414153 0.90 STAT6 (0.38) ALDH1A1NPSR1CYP1A2CYP3A4GAA
SCHEMBL6414138 0.90 STAT6 (0.38) ALDH1A1NPSR1CYP1A2CYP3A4GAA
SCHEMBL6419260 0.88 PHGDH (0.40) ALDH1A1POLBHPGDHSD17B10CTDSP1
SCHEMBL6413677 0.87 KDM5B (0.42) ALDH1A1POLBHPGDHSD17B10CTDSP1
SCHEMBL6413651 0.87 KDM5B (0.42) ALDH1A1POLBHPGDHSD17B10CTDSP1
SCHEMBL6413574 0.83 GSK3B (0.40) CSNK2A1MEN1MAPTKMT2AKDM4E
SCHEMBL6413560 0.83 GSK3B (0.40) CSNK2A1MEN1MAPTKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050143382-A1 Heterocyclic compounds as pharmaceutically active compounds 4SC AG (DE) 2005-06-30 US disclosed
WO-2005044270-A1 OXADIAZOLOPYRAZINE DERIVATIVES AS PHARMACEUTICALLY ACTIVE COMPOUNDS 4SC AG (DE) 2005-05-19 WO disclosed
EP-1529531-A1 Oxadiazolopyrazine derivatives as pharmaceutically active compounds 4SC AG (DE) 2005-05-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050143382-A1 Heterocyclic compounds as pharmaceutically active compounds NR5A2, NR1H2, NR2C2 ALDH1A1 1119/4885POLB 3589/4885HPGD 2524/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.