SCHEMBL6433711

SCHEMBL6433711

CC(C)CNC(=O)OC1=NOC2(CCN(C(=O)c3cccc4ccccc34)CC2)C1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 1/20 0.43
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
ALDH1A1 P00352 3/20 0.40
LMNA P02545 1/20 0.40
CCR5 P51681 2/20 0.40
POLB P06746 1/20 0.40
HTT P42858 1/20 0.40
TGM2 P21980 4/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CHRM2 P08172 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2399133 0.85 AVPR1A (0.45) AVPR1AJAK2JAK1ALDH1A1LMNA
SCHEMBL6415557 0.84 KMT2A (0.45) ALDH1A1LMNAMEN1KMT2A
SCHEMBL6431092 0.84 AVPR1A (0.41) AVPR1AJAK2JAK1ALDH1A1LMNA
SCHEMBL6410357 0.80 POLB (0.43) ALDH1A1LMNAPOLBHTT
SCHEMBL6411397 0.78 ALDH1A1 (0.42) ALDH1A1LMNAHTTMEN1KMT2A
SCHEMBL6409874 0.77 FASN (0.40) KMT2A
SCHEMBL6413248 0.74 AVPR1A (0.54) AVPR1AJAK2JAK1ALDH1A1LMNA
SCHEMBL6410188 0.73 MEN1 (0.45) ALDH1A1LMNAHTTMEN1KMT2A
SCHEMBL6410103 0.73 CYP2D6 (0.42) ALDH1A1MEN1KMT2A
SCHEMBL6410008 0.72 DRD2 (0.39) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401841-B1 SUBSTITUTED 1-OXA-2,8-DIAZA-SPIRO 4,5]DEC-2-ENE DERIVATIVES AS MEDICAMENTS FOR THE TREATMENT OF PAIN GRUENENTHAL GMBH (DE) 2005-08-24 EP disclosed