Ethylene

Ethylene

SCHEMBL6433762

C=C.CC(C)S(=O)(=O)N1CCC(=O)CC1

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.38
CYP3A4 P08684 1/20 0.37
CYP3A5 P20815 1/20 0.37
EPHX2 P34913 2/20 0.35
GRM5 P41594 1/20 0.33
ALDH1A1 P00352 1/20 0.32
NAMPT P43490 2/20 0.31
CYP17A1 P05093 1/20 0.31
CYP21A2 P08686 1/20 0.31
CYP11B1 P15538 1/20 0.31
PARP1 P09874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12251515 0.96 KMT2A (0.40) KMT2ACYP3A4CYP3A5EPHX2GRM5
SCHEMBL17631813 0.88 EPHX2 (0.36) KMT2ACYP3A4CYP3A5EPHX2GRM5
SCHEMBL18638767 0.79 KMT2A (0.38) KMT2A
SCHEMBL13100462 0.77
Ethylene SCHEMBL6434698 0.76 KMT2A (0.41) KMT2ACYP3A4ALDH1A1
SCHEMBL16022965 0.72 EPHX2 (0.44) KMT2ACYP3A4CYP3A5EPHX2ALDH1A1
SCHEMBL5405216 0.72 EPHX2 (0.44) KMT2ACYP3A4EPHX2ALDH1A1
SCHEMBL17644092 0.72 EPHX2 (0.40) KMT2AEPHX2GRM5
SCHEMBL3741198 0.71 EPHX2 (0.38) KMT2ACYP3A4CYP3A5EPHX2ALDH1A1
SCHEMBL17631926 0.71 EPHX2 (0.39) KMT2AEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050026836-A1 Composition for the treatment of damaged tissue DACK KEVIN NEIL (GB) 2005-02-03 US disclosed
US-20030199440-A1 Composition for the treatment of damaged tissue PFIZER INC. 2003-10-23 US disclosed
EP-1181017-B1 METALLOPROTEASE INHIBITORS PFIZER LTD (GB) 2003-04-16 EP disclosed
US-6511993-B1 Substituted alpha-aminosulphonyl-acetohydroxamic acids which are inhibitors of zinc-dependent metalloprotease enzymes PFIZER INC. 2003-01-28 US disclosed
EP-1242120-A2 COMBINATIONS OF GROWTH FACTORS AND I:UPA OR I:MMP FOR THE TREATMENT OF DAMAGED TISSUE Pfizer Limited (GB) 2002-09-25 EP disclosed
EP-1181017-A1 METALLOPROTEASE INHIBITORS Pfizer Limited (GB) 2002-02-27 EP disclosed
WO-2001049309-A2 COMBINATIONS OF GROWTH FACTORS AND I: UPA OR I: MMP FOR THE TREATMENT OF DAMAGED TISSUE PFIZER LIMITED (GB) 2001-07-12 WO disclosed
WO-2000074681-A1 METALLOPROTEASE INHIBITORS PFIZER LIMITED (GB) 2000-12-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030199440-A1 Composition for the treatment of damaged tissue MMP1, SERPINE1, COL14A1 KMT2A 4810/4885CYP3A4 4668/4885CYP3A5 4497/4885
US-20050026836-A1 Composition for the treatment of damaged tissue MMP1, SERPINE1, COL14A1 KMT2A 4810/4885CYP3A4 4668/4885CYP3A5 4497/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.