SCHEMBL6434684

SCHEMBL6434684

Cc1cccc(N)c1-c1nc[nH]n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD44 P16070 1/20 0.41
CYP3A4 P08684 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
DPP4 P27487 1/20 0.36
GAA P10253 2/20 0.36
TSHR P16473 1/20 0.35
PIK3CA P42336 1/20 0.35
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
MAPT P10636 1/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
POLB P06746 1/20 0.31
APOBEC3G Q9HC16 1/20 0.31
SRC P12931 1/20 0.31
KEAP1 Q14145 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
PARP1 P09874 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3279505 0.81 MAP4K1 (0.40) GAANPC1
SCHEMBL6434686 0.77 PIK3CA (0.43) CD44CYP3A4TDP1GAATSHR
SCHEMBL30839716 0.76 CD44 (0.65) CD44CYP3A4TDP1DPP4TSHR
SCHEMBL3462069 0.76 CD44 (0.65) CD44CYP3A4TDP1DPP4TSHR
SCHEMBL11686059 0.72 IDO1 (0.52) CYP3A4TDP1GAAMAPTKDM4E
SCHEMBL15125436 0.72 GAA (0.52) CYP3A4GAATSHRPIK3CAKDM4E
SCHEMBL15942236 0.70 TSHR (0.43) CYP3A4TDP1TSHRMAPTKDM4E
SCHEMBL17194909 0.70 BRD4 (0.36) CYP3A4GAATSHRMAPTKDM4E
SCHEMBL10726692 0.70 ALDH1A1 (0.53) CYP3A4TDP1TSHRMAPTKDM4E
SCHEMBL16497559 0.69 CD44 (0.62) CD44CYP3A4TDP1DPP4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050288347-A1 Certain triazole-based compounds, compositions, and uses thereof AGRIUS GROUP, LLC. 2005-12-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050288347-A1 Certain triazole-based compounds, compositions, and uses thereof ABCG2, ATP5ME, DNTT CD44 4393/4885CYP3A4 25/4885TDP1 288/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.