SCHEMBL6434747

SCHEMBL6434747

CC(C)(C)OC(=O)CNc1ccc(N)cn1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 1/20 0.41
PTGS1 P23219 3/20 0.41
FTO Q9C0B1 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
KDM5B Q9UGL1 1/20 0.38
KDM2A Q9Y2K7 1/20 0.38
KDM3A Q9Y4C1 1/20 0.38
HCAR3 P49019 3/20 0.37
PPIB P23284 1/20 0.35
PPIA P62937 1/20 0.35
PPID Q08752 1/20 0.35
PPIG Q13427 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAPK8 P45983 1/20 0.35
MAP4K4 O95819 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18286138 0.83 PTK2 (0.49) CCNT1ALDH1A1L3MBTL1
SCHEMBL12295518 0.83 RAB9A (0.45) CCNT1ALDH1A1
SCHEMBL31407474 0.83 RAB9A (0.45) CCNT1ALDH1A1
SCHEMBL691502 0.82 HCAR3 (0.60) HCAR3
SCHEMBL2068741 0.81 CCNT1 (0.42) CCNT1HCAR3KDM4EALDH1A1L3MBTL1
SCHEMBL30980609 0.80 CRBN (0.41) PTGS1HCAR3KDM4EALDH1A1
SCHEMBL1724626 0.80 DPP4 (0.47) CCNT1
SCHEMBL1725418 0.79 HCAR3 (0.41) CCNT1HCAR3
SCHEMBL15905735 0.79 HCAR3 (0.41) CCNT1HCAR3
SCHEMBL1725419 0.79 HCAR3 (0.41) CCNT1HCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040111-B1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2005-06-22 EP disclosed
US-6268378-B1 TREATING AND PREVENTING OSTEOPOROSIS, AND INHIBITING VASCULAR RESTENOSIS, DIABETIC RETINOPATHY, MACULAR DEGENERATION, ANGIOGENESIS, ATHEROSCLEROSIS, INFLAMMATION, VIRAL DISEASE, AND TUMOR GROWTH. MERCK & CO., INC. 2001-07-31 US disclosed
US-6066648-A USEFUL IN INHIBITING BONE RESORPTION, TREATING AND PREVENTING OSTEOPOROSIS, AND INHIBITING VASCULAR RESTENOSIS, DIABETIC RETINOPATHY, MACULAR DEGENERATION, ANGIOGENESIS, ATHEROSCLEROSIS, INFLAMMATION, VIRAL DISEASE, AND TUMOR GROWTH MERCK & CO., INC. (US) 2000-05-23 US disclosed
US-6017926-A Integrin receptor antagonists MERCK & CO., INC. (US) 2000-01-25 US disclosed