SCHEMBL6436867

SCHEMBL6436867

COc1ccc(C(=O)c2ccc(OC)c(I)c2)cc1I

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.68
CYP2C19 P33261 2/20 0.68
CYP3A4 P08684 1/20 0.68
CYP2C9 P11712 1/20 0.68
TSHR P16473 1/20 0.68
ALDH1A1 P00352 3/20 0.61
HTT P42858 3/20 0.61
LMNA P02545 2/20 0.61
L3MBTL1 Q9Y468 1/20 0.61
SLC22A6 Q4U2R8 1/20 0.58
SLC22A8 Q8TCC7 1/20 0.58
GAA P10253 1/20 0.58
TUBB4A P04350 3/20 0.53
TUBB P07437 3/20 0.53
TUBA3C P0DPH7 3/20 0.53
TUBA1B P68363 3/20 0.53
TUBA4A P68366 3/20 0.53
TUBB4B P68371 3/20 0.53
TUBB3 Q13509 3/20 0.53
TUBB2A Q13885 3/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6437851 0.91 ALDH1A1 (0.73) CYP1A2CYP2C19CYP3A4CYP2C9TSHR
SCHEMBL12635170 0.90 TUBB4A (0.69) CYP1A2CYP2C19CYP3A4CYP2C9TSHR
SCHEMBL16185983 0.87 CYP1A2 (0.53) CYP1A2CYP2C19CYP3A4CYP2C9TSHR
SCHEMBL7943307 0.86 ALDH1A1 (0.54) CYP1A2CYP2C19CYP3A4CYP2C9TSHR
SCHEMBL787550 0.86 TPMT (0.69) CYP1A2CYP2C19CYP3A4CYP2C9TSHR
SCHEMBL30010958 0.86 TPMT (0.69) CYP1A2CYP2C19CYP3A4CYP2C9TSHR
SCHEMBL12574135 0.86 CYP1A2 (0.56) CYP1A2CYP2C19CYP3A4CYP2C9TSHR
SCHEMBL29375569 0.85 MAPK1 (0.58) CYP1A2CYP2C19CYP3A4CYP2C9TSHR
SCHEMBL31704508 0.85 MAPT (0.62) CYP1A2CYP2C19CYP3A4CYP2C9TSHR
SCHEMBL29375601 0.85 TSHR (0.48) CYP1A2CYP2C19CYP3A4CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106459062-A Substituted [1,2,4] triazolo [1,5-a ] pyrimidin-7-yl compounds as PDE2 inhibitors 达特神经科学(开曼)有限公司 2017-02-22 CN disclosed
CN-106065010-A For treating or prevent the compound of hyperuricemia or gout 镇江新元素医药科技有限公司 2016-11-02 CN disclosed
EP-1506959-A2 Derivatised molecules for mass spectrometry OXFORD GENE TECHNOLOGY IP LIMITED (GB) 2005-02-16 EP disclosed