SCHEMBL6437304

SCHEMBL6437304

CC(C)(C)OC(=O)N(CC=O)C[C@@H](O[Si](C)(C)C(C)(C)C)c1cccc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.36
CPB2 Q96IY4 1/20 0.32
MDM2 Q00987 8/20 0.32
TP53 P04637 7/20 0.32
S1PR3 Q99500 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GRM5 P41594 1/20 0.32
ITGB1 P05556 1/20 0.32
ITGA4 P13612 1/20 0.32
BACE1 P56817 1/20 0.32
XPO1 O14980 1/20 0.32
SLC6A2 P23975 3/20 0.31
SLC6A4 P31645 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5949847 1.00 AOC3 (0.36) AOC3CPB2MDM2TP53S1PR3
SCHEMBL5949849 1.00 AOC3 (0.36) AOC3CPB2MDM2TP53S1PR3
SCHEMBL5950226 0.90 AOC3 (0.35) AOC3CPB2S1PR3SMN1; SMN2BACE1
SCHEMBL6435807 0.90 APP (0.32)
SCHEMBL6435801 0.90 APP (0.32)
SCHEMBL7977761 0.89 AOC3 (0.35) AOC3CPB2S1PR3BACE1XPO1
SCHEMBL7716940 0.85 AOC3 (0.38) AOC3S1PR3BACE1
SCHEMBL7716942 0.85 AOC3 (0.38) AOC3S1PR3BACE1
SCHEMBL9267480 0.84 AOC3 (0.36) AOC3S1PR3ITGB1ITGA4BACE1
SCHEMBL7716904 0.84 AOC3 (0.36) AOC3CPB2S1PR3BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1087943-B1 THERAPEUTIC BIARYL DERIVATIVES GLAXO GROUP LTD (GB) 2005-08-17 EP disclosed
US-6251925-B1 AN AGONISTS FOR HUMAN BETA-3 ADRENOCEPTOR GLAXO WELLCOME INC. 2001-06-26 US disclosed
EP-1087943-A1 THERAPEUTIC BIARYL DERIVATIVES GLAXO GROUP LIMITED (GB) 2001-04-04 EP disclosed
WO-1999065877-A1 THERAPEUTIC BIARYL DERIVATIVES GLAXO GROUP LIMITED (GB) 1999-12-23 WO disclosed