SCHEMBL7716904

SCHEMBL7716904

COC(=O)CCN(C[C@@H](O[Si](C)(C)C(C)(C)C)c1cccc(Cl)c1)C(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.36
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
FDFT1 P37268 1/20 0.33
GLS O94925 1/20 0.33
S1PR3 Q99500 1/20 0.33
CASR P41180 1/20 0.33
IDO1 P14902 1/20 0.32
ADRB3 P13945 2/20 0.32
BACE1 P56817 1/20 0.32
WDR5 P61964 1/20 0.32
GLA P06280 1/20 0.32
ADRB2 P07550 1/20 0.32
ADRB1 P08588 1/20 0.32
PNP P00491 1/20 0.32
CTSL P07711 1/20 0.31
CPB2 Q96IY4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7716942 0.91 AOC3 (0.38) AOC3S1PR3CASRADRB3BACE1
SCHEMBL7716940 0.91 AOC3 (0.38) AOC3S1PR3CASRADRB3BACE1
SCHEMBL5950226 0.86 AOC3 (0.35) AOC3S1PR3ADRB3BACE1CPB2
SCHEMBL5949849 0.84 AOC3 (0.36) AOC3S1PR3BACE1CPB2
SCHEMBL5949847 0.84 AOC3 (0.36) AOC3S1PR3BACE1CPB2
SCHEMBL6437304 0.84 AOC3 (0.36) AOC3S1PR3BACE1CPB2
SCHEMBL4474573 0.83 ADRB3 (0.39) AOC3MEN1KMT2AADRB3BACE1
SCHEMBL4474577 0.83 ADRB3 (0.39) AOC3MEN1KMT2AADRB3BACE1
SCHEMBL7714567 0.82 ADRB2 (0.31) ADRB3ADRB2ADRB1
SCHEMBL8100555 0.82 ADRB2 (0.31) ADRB3ADRB2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865421-B1 ARYLETHANOLAMINE DERIVATIVES AND THEIR USE AS AGONISTS OF ATYPICAL BETA-ADRENOCEPTORS GLAXO GROUP LTD (GB) 2002-03-27 EP disclosed