SCHEMBL7716940

SCHEMBL7716940

COC(=O)CN(CC(O[Si](C)(C)C(C)(C)C)c1cccc(Cl)c1)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.38
CASR P41180 1/20 0.35
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
S1PR3 Q99500 1/20 0.33
BACE1 P56817 3/20 0.33
WDR5 P61964 1/20 0.33
GLA P06280 1/20 0.33
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
ADRB3 P13945 1/20 0.33
PNP P00491 1/20 0.33
CCR5 P51681 1/20 0.32
CTSL P07711 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7716942 1.00 AOC3 (0.38) AOC3CASRNPC1RAB9AS1PR3
SCHEMBL7716904 0.91 AOC3 (0.36) AOC3CASRS1PR3BACE1WDR5
SCHEMBL7977761 0.88 AOC3 (0.35) AOC3S1PR3BACE1
SCHEMBL5949847 0.85 AOC3 (0.36) AOC3S1PR3BACE1
SCHEMBL5949849 0.85 AOC3 (0.36) AOC3S1PR3BACE1
SCHEMBL6437304 0.85 AOC3 (0.36) AOC3S1PR3BACE1
SCHEMBL5950226 0.84 AOC3 (0.35) AOC3S1PR3BACE1ADRB3
SCHEMBL4474577 0.81 ADRB3 (0.39) AOC3BACE1ADRB1ADRB3
SCHEMBL4474573 0.81 ADRB3 (0.39) AOC3BACE1ADRB1ADRB3
SCHEMBL7714567 0.81 ADRB2 (0.31) ADRB2ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865421-B1 ARYLETHANOLAMINE DERIVATIVES AND THEIR USE AS AGONISTS OF ATYPICAL BETA-ADRENOCEPTORS GLAXO GROUP LTD (GB) 2002-03-27 EP disclosed
US-6048872-A DIETETICS; ANTIDIABETIC AGENTS; CARDIOVASCULAR DISORDERS; GASTROINTESTINAL DISORDERS GLAXO WELLCOME INC. (US) 2000-04-11 US disclosed
WO-1995033724-A1 PHENETHANOLAMINE DERIVATIVES AND THEIR USE AS ATYPICAL BETA-ADRENOCEPTOR AGONISTS GLAXO GROUP LIMITED (GB) 1995-12-14 WO disclosed