SCHEMBL6437855

SCHEMBL6437855

Cc1nn(CC(=O)Nc2sc3c(c2C(=O)O)CCCC3)c(C)c1[N+](=O)[O-]

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.58
MAPT P10636 2/20 0.58
GAA P10253 2/20 0.58
HPGD P15428 2/20 0.57
HTT P42858 3/20 0.52
POLB P06746 1/20 0.52
LMNA P02545 2/20 0.51
NPC1 O15118 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3918756 0.91 ALDH1A1 (0.70) ALDH1A1MAPTGAAHPGDHTT
SCHEMBL3921443 0.91 GAA (0.63) ALDH1A1MAPTGAAHPGDHTT
SCHEMBL3914838 0.87 GAA (0.76) ALDH1A1MAPTGAAHPGDHTT
SCHEMBL3278975 0.85 ALDH1A1 (0.78) ALDH1A1MAPTGAAHPGDHTT
SCHEMBL8289416 0.80 ALDH1A1 (0.60) ALDH1A1MAPTGAAHPGDPOLB
SCHEMBL3916269 0.76 CYP1A2 (0.77) ALDH1A1MAPTGAAHPGDHTT
SCHEMBL3922647 0.76 MAPT (0.59) ALDH1A1MAPTGAAHPGDHTT
SCHEMBL3914074 0.76 CYP1A2 (0.54) ALDH1A1MAPTGAAHPGDHTT
SCHEMBL681864 0.75 ALDH1A1 (0.80) ALDH1A1MAPTHTTPOLBLMNA
SCHEMBL6437411 0.73 ALDH1A1 (0.77) ALDH1A1MAPTGAAHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1492783-A1 4,5,6,7-TRETRAHYDROBENZO(B) THIOPHENE DERIVATIVES AND METHODS FOR MEDICAL INTERVENTION AGAINST MYCROBACTERIAL INFECTIONS Axxima Pharmaceuticals AG (DE) 2005-01-05 EP claimed
WO-2003084947-A1 4,5,6,7-TRETRAHYDROBENZO[B] THIOPHENE DERIVATIVES AND METHODS FOR MEDICAL INTERVENTION AGAINST MYCROBACTERIAL INFECTIONS AXXIMA PHARMACEUTICALS AG (DE) 2003-10-16 WO claimed