SCHEMBL6438770

SCHEMBL6438770

C=CCC(=CBr)c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.39
HDAC1 Q13547 2/20 0.37
HDAC2 Q92769 2/20 0.37
HDAC3 O15379 1/20 0.37
NCOR2 Q9Y618 1/20 0.37
MAOA P21397 2/20 0.36
MAOB P27338 2/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
PTPN1 P18031 1/20 0.34
GSK3B P49841 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11673299 0.81 AKT1 (0.40) AKT1HDAC1HDAC2HDAC3NCOR2
SCHEMBL9596280 0.81 AKT1 (0.40) AKT1HDAC1HDAC2HDAC3NCOR2
SCHEMBL11673293 0.81 AKT1 (0.40) AKT1HDAC1HDAC2HDAC3NCOR2
SCHEMBL1076032 0.81 AKT1 (0.40) AKT1HDAC1HDAC2HDAC3NCOR2
SCHEMBL11048295 0.79 AKT1 (0.39) AKT1HDAC1HDAC2HDAC3NCOR2
SCHEMBL476634 0.79 MAOA (0.53) AKT1HDAC1HDAC2HDAC3NCOR2
SCHEMBL727277 0.79 AKT1 (0.39) AKT1HDAC1HDAC2HDAC3NCOR2
SCHEMBL1076558 0.79 MAOA (0.40) AKT1HDAC1HDAC2HDAC3NCOR2
SCHEMBL9723351 0.79 AKT1 (0.39) AKT1HDAC1HDAC2HDAC3NCOR2
SCHEMBL11048275 0.79 AKT1 (0.39) AKT1HDAC1HDAC2HDAC3NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3541635-B1 TIRE COMPRISING A BLOCK COPOLYMER COMPRISING AN ELASTOMERIC BLOCK HAVING UNITS OF ISOBUTYLENE AND HALOGENOALKYLSTYRENE MICHELIN & CIE (FR) 2020-12-30 EP claimed
EP-3541635-A1 PNEUMATIC TYRE COMPRISING A BLOCK COPOLYMER COMPRISING AN ELASTOMER BLOCK WITH ISOBUTYLENE AND HALOGENOALKYL STYRENE UNITS Compagnie Générale des Etablissements Michelin (FR) 2019-09-25 EP claimed
US-6837288-B2 Composition for tire sidewalls and other rubber constructions EXXONMOBIL CHEMICAL PATENTS INC. (US) 2005-01-04 US claimed
EP-0981581-B1 COMPOSITION FOR TIRE SIDEWALLS AND OTHER RUBBER CONSTRUCTIONS EXXONMOBIL CHEM PATENTS INC (US) 2002-12-11 EP claimed
US-20020100530-A1 Composition for tire sidewalls and other rubber constructions HOLLEY PERFORMANCE PRODUCTS INC. 2002-08-01 US claimed
US-6374889-B1 RUBBER BLENDS OF BROMINATED ISOBUTYLENE/PARA-METHYLSTYRENE COPOLYMERS; GOOD CURE CHARACTERISTICS, GOOD ADHESION AND FLEX CRACK RESISTANCE, AS WELL AS OZONE RESISTANCE. EXXONMOBIL CHEMICAL PATENTS INC. 2002-04-23 US claimed
JP-2002512652-A 2002-04-23 JP claimed
EP-0981581-A1 COMPOSITION FOR TIRE SIDEWALLS AND OTHER RUBBER CONSTRUCTIONS EXXON CHEMICAL PATENTS INC. (US) 2000-03-01 EP claimed
WO-1998050464-A1 COMPOSITION FOR TIRE SIDEWALLS AND OTHER RUBBER CONSTRUCTIONS EXXON CHEMICAL PATENTS INC. (US) 1998-11-12 WO claimed
CN-115960291-A Preparation method of long-chain haloalkyl styrene polymer 南京大学 2023-04-14 CN disclosed
US-11597189-B2 Refrigerant-transporting hose THE YOKOHAMA RUBBER CO., LTD. (JP) 2023-03-07 US disclosed
US-20210162722-A1 REFRIGERANT-TRANSPORTING HOSE THE YOKOHAMA RUBBER CO., LTD. (JP) 2021-06-03 US disclosed
EP-3541635-B1 TIRE COMPRISING A BLOCK COPOLYMER COMPRISING AN ELASTOMERIC BLOCK HAVING UNITS OF ISOBUTYLENE AND HALOGENOALKYLSTYRENE MICHELIN & CIE (FR) 2020-12-30 EP disclosed
EP-3541635-A1 PNEUMATIC TYRE COMPRISING A BLOCK COPOLYMER COMPRISING AN ELASTOMER BLOCK WITH ISOBUTYLENE AND HALOGENOALKYL STYRENE UNITS Compagnie Générale des Etablissements Michelin (FR) 2019-09-25 EP disclosed
EP-0981581-B1 COMPOSITION FOR TIRE SIDEWALLS AND OTHER RUBBER CONSTRUCTIONS EXXONMOBIL CHEM PATENTS INC (US) 2002-12-11 EP disclosed
US-20020100530-A1 Composition for tire sidewalls and other rubber constructions HOLLEY PERFORMANCE PRODUCTS INC. 2002-08-01 US disclosed
US-6374889-B1 RUBBER BLENDS OF BROMINATED ISOBUTYLENE/PARA-METHYLSTYRENE COPOLYMERS; GOOD CURE CHARACTERISTICS, GOOD ADHESION AND FLEX CRACK RESISTANCE, AS WELL AS OZONE RESISTANCE. EXXONMOBIL CHEMICAL PATENTS INC. 2002-04-23 US disclosed
EP-0981581-A1 COMPOSITION FOR TIRE SIDEWALLS AND OTHER RUBBER CONSTRUCTIONS EXXON CHEMICAL PATENTS INC. (US) 2000-03-01 EP disclosed
US-6025447-A Graft copolymers BASF AKTIENGESELLSCHAFT (DE) 2000-02-15 US disclosed
WO-1998050464-A1 COMPOSITION FOR TIRE SIDEWALLS AND OTHER RUBBER CONSTRUCTIONS EXXON CHEMICAL PATENTS INC. (US) 1998-11-12 WO disclosed