SCHEMBL6439703

SCHEMBL6439703

CS(=O)(=O)c1ccc(-c2[nH]nc(COc3cccc(CBr)c3)c2C2CCCCC2)cc1

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.37
PPARG P37231 3/20 0.35
PPARA Q07869 3/20 0.35
PTGS1 P23219 2/20 0.34
F10 P00742 1/20 0.34
GHSR Q92847 1/20 0.33
VCP P55072 1/20 0.33
AKT1 P31749 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6438974 0.91 KDR (0.39) PTGS2PPARGPPARAPTGS1F10
SCHEMBL6438455 0.89 PTGS2 (0.43) PTGS2PPARGPPARAPTGS1F10
SCHEMBL6442228 0.82 PTGS2 (0.44) PTGS2PTGS1GHSR
SCHEMBL6439880 0.77 PTGS2 (0.49) PTGS2PTGS1GHSR
SCHEMBL6441485 0.76 PTGS2 (0.41) PTGS2PTGS1GHSR
SCHEMBL6438872 0.76 PTGS2 (0.47) PTGS2PTGS1GHSR
SCHEMBL6439597 0.75 PTGS2 (0.41) PTGS2PTGS1GHSR
SCHEMBL6438496 0.73 PTGS2 (0.43) PTGS2PTGS1GHSR
SCHEMBL6527042 0.73 PTGS2 (0.45) PTGS2PTGS1
SCHEMBL3869384 0.73 PTGS2 (0.64) PTGS2PTGS1VCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP disclosed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP disclosed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed