SCHEMBL6440067

SCHEMBL6440067

COc1ccc(-c2c(COCCCO[N+](=O)[O-])n[nH]c2-c2ccc(S(C)(=O)=O)cc2)cc1[N+](=O)[O-]

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 1/20 0.39
PDGFRA P16234 1/20 0.39
PTGS2 P35354 8/20 0.38
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
GRK6 P43250 1/20 0.38
PTGS1 P23219 1/20 0.36
FYN P06241 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
CASP6 P55212 1/20 0.34
CTDSP1 Q9GZU7 1/20 0.34
AGTR1 P30556 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6522743 0.86 PTGS2 (0.45) PTGS2PTGS1
SCHEMBL6441194 0.84 PTGS2 (0.46) PTGS2PTGS1
SCHEMBL6440855 0.84 PTGS2 (0.42) PTGS2PTGS1
SCHEMBL6438240 0.83 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL6441773 0.83 PTGS2 (0.40) PTGS2PTGS1
SCHEMBL6441366 0.80 PTGS2 (0.39) PTGS2
SCHEMBL3863757 0.77 CA1 (0.46) PTGS2ALDH1A1PTGS1
SCHEMBL3864964 0.75 CA12 (0.46) PTGS2PTGS1
SCHEMBL6527042 0.74 PTGS2 (0.45) PTGS2PTGS1
SCHEMBL3867384 0.73 PTGS2 (0.52) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP disclosed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP disclosed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed