SCHEMBL6438240

SCHEMBL6438240

CS(=O)(=O)c1ccc(-c2[nH]nc(COCCCO[N+](=O)[O-])c2-c2ccc(F)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.48
ESR2 Q92731 1/20 0.45
PTGS1 P23219 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6440855 0.91 PTGS2 (0.42) PTGS2ESR2PTGS1
SCHEMBL6441194 0.91 PTGS2 (0.46) PTGS2ESR2PTGS1
SCHEMBL6441773 0.90 PTGS2 (0.40) PTGS2ESR2PTGS1
SCHEMBL6441366 0.90 PTGS2 (0.39) PTGS2ESR2
SCHEMBL6522743 0.89 PTGS2 (0.45) PTGS2ESR2PTGS1
SCHEMBL3863757 0.83 CA1 (0.46) PTGS2PTGS1
SCHEMBL6440067 0.83 PDGFRB (0.39) PTGS2PTGS1
SCHEMBL3864105 0.82 CA12 (0.46) PTGS2PTGS1
SCHEMBL3864964 0.82 CA12 (0.46) PTGS2PTGS1
SCHEMBL6440170 0.80 ESR2 (0.49) PTGS2ESR2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP claimed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP claimed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO claimed
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP disclosed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP disclosed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed