SCHEMBL6440085

SCHEMBL6440085

O=C1CC=[C]c2ccccc2N1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.42
PDK2 Q15119 1/20 0.42
PLCG1 P19174 1/20 0.42
NPC1 O15118 1/20 0.41
MAPK13 O15264 1/20 0.41
MAPK12 P53778 1/20 0.41
MAPK11 Q15759 1/20 0.41
MAPK14 Q16539 1/20 0.41
MAPT P10636 2/20 0.39
ALDH1A1 P00352 4/20 0.38
BRD4 O60885 7/20 0.37
CREBBP Q92793 7/20 0.37
EP300 Q09472 1/20 0.37
EPHX2 P34913 1/20 0.36
TSHR P16473 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HSD17B10 Q99714 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1973489 0.72 AHR (0.45) AHRPDK2PLCG1NPC1MAPK13
SCHEMBL6441774 0.69 NPC1 (0.50) AHRPDK2PLCG1NPC1MAPK13
SCHEMBL2519570 0.68 GABRA1 (0.42) AHRPDK2PLCG1NPC1MAPK13
SCHEMBL151990 0.67 GAA (0.31) HSD17B10
SCHEMBL1973487 0.65 AHR (0.47) AHRPDK2PLCG1NPC1MAPK13
SCHEMBL6379887 0.65 AHR (0.70) AHRPDK2PLCG1NPC1MAPK13
SCHEMBL1235044 0.65 AHR (0.70) AHRPDK2PLCG1NPC1MAPK13
SCHEMBL29510715 0.65 AHR (0.70) AHRPDK2PLCG1NPC1MAPK13
SCHEMBL302509 0.64 MAOA (0.37) AHRPDK2PLCG1NPC1MAPK13
SCHEMBL29246 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1286673-B8 LIGANDS OF INTEGRIN RECEPTORS ABBOTT GMBH & CO KG (DE) 2005-07-20 EP disclosed
EP-1286673-A2 LIGANDS OF INTEGRIN RECEPTORS Basf Aktiengesellschaft (DE) 2003-03-05 EP disclosed
WO-2001093840-A2 LIGANDS OF INTEGRIN RECEPTORS BASF AG (DE) 2001-12-13 WO disclosed