SCHEMBL6440982

SCHEMBL6440982

CS(=O)(=O)NC(=O)C(c1ccc(OCc2ccc3ccccc3n2)cc1)C1CCCCCC1

nearest known ligand 0.73

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 20/20 0.73
HDAC6 Q9UBN7 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30209466 1.00 ALOX5 (0.73) ALOX5HDAC6
SCHEMBL6440984 1.00 ALOX5 (0.73) ALOX5HDAC6
SCHEMBL8892800 0.89 ALOX5 (0.78) ALOX5HDAC6
SCHEMBL9315247 0.88 ALOX5 (0.80) ALOX5HDAC6
SCHEMBL9303393 0.87 ALOX5 (0.75) ALOX5HDAC6
SCHEMBL8895036 0.87 ALOX5 (0.75) ALOX5HDAC6
SCHEMBL9301897 0.86 ALOX5 (0.77) ALOX5HDAC6
SCHEMBL8892164 0.86 ALOX5 (0.75) ALOX5HDAC6
SCHEMBL9431826 0.86 ALOX5 (0.80) ALOX5HDAC6
SCHEMBL8827857 0.86 ALOX5 (0.80) ALOX5HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0637961-A4 METHODS FOR TREATING INFLAMMATORY BOWEL DISEASE WITH LEUKOTRIENE SYNTHESIS INHIBITORS. MILES INC (US) 1995-08-09 EP claimed
EP-0637961-A1 METHODS FOR TREATING INFLAMMATORY BOWEL DISEASE WITH LEUKOTRIENE SYNTHESIS INHIBITORS Bayer Corporation (US) 1995-02-15 EP claimed
WO-1994018976-A1 METHODS FOR TREATING INFLAMMATORY BOWEL DISEASE WITH LEUKOTRIENE SYNTHESIS INHIBITORS MILES INC. (US) 1994-09-01 WO claimed
JP-6192228-A None JP disclosed
JP-6192228-A None JP disclosed
US-20050222193-A1 Novel combination for the treatment of airway disorders ALTANA PHARMA AG (DE) 2005-10-06 US disclosed
WO-2005074932-A1 THE USE OF (S) - PANTOPRAZOLE MAGNESIUM FOR THE TREATMENT OF AIRWAY DISORDERS ALTANA PHARMA AG (DE) 2005-08-18 WO disclosed
US-20050165041-A1 Combination for the treatment of airway disorders ALTANA PHARMA AG (DE) 2005-07-28 US disclosed
EP-1517706-A2 COMBINATION OF A PROTON PUMP INHIBITOR AND A RESPIRATORY AGENT FOR THE TREATMENT OF RESPIRATORY DISEASES ALTANA Pharma AG (DE) 2005-03-30 EP disclosed
EP-1506016-A2 NEW COMBINATION OF REVERSIBLE PROTON PUMP INHIBITORS AND AIRWAY THERAPEUTICS FOR TREATING AIRWAY DISORDERS ALTANA Pharma AG (DE) 2005-02-16 EP disclosed
WO-2003094967-A2 NEW COMBINATION OF REVERSIBLE PROTON PUMP INHIBITORS AND AIRWAY THERAPEUTICS FOR TREATING AIRWAY DISORDERS ALTANA PHARMA AG (DE) 2003-11-20 WO disclosed
WO-2003094968-A2 COMBINATION OF A PROTON PUMP INHIBITOR AND A RESPIRATORY AGENT FOR THE TREATMENT OF RESPIRATORY DISEASES ALTANA PHARMA AG (DE) 2003-11-20 WO disclosed
EP-0637961-A4 METHODS FOR TREATING INFLAMMATORY BOWEL DISEASE WITH LEUKOTRIENE SYNTHESIS INHIBITORS. MILES INC (US) 1995-08-09 EP disclosed
US-5391555-A Administering 2-(4(2-quinolinyl-methoxy)-phenyl)-acetic acid derivatives; Crohn's disease MILES INC. (US) 1995-02-21 US disclosed
EP-0637961-A1 METHODS FOR TREATING INFLAMMATORY BOWEL DISEASE WITH LEUKOTRIENE SYNTHESIS INHIBITORS Bayer Corporation (US) 1995-02-15 EP disclosed
WO-1994018976-A1 METHODS FOR TREATING INFLAMMATORY BOWEL DISEASE WITH LEUKOTRIENE SYNTHESIS INHIBITORS MILES INC. (US) 1994-09-01 WO disclosed
JP-H06192228-A CRYSTALLINE (R)-(-)-2-XYCLOHEPTYL-N-METHYLSULFONYL-(4-(2-QUINOLINYLMETHOXY)-PHENYL)-ACETOAMIDE BAYER AG 1994-07-12 JP disclosed
JP-H06192228-A CRYSTALLINE (R)-(-)-2-XYCLOHEPTYL-N-METHYLSULFONYL-(4-(2-QUINOLINYLMETHOXY)-PHENYL)-ACETOAMIDE BAYER AG 1994-07-12 JP disclosed
EP-0593976-A1 Crystalline (R)-(-)-2-cycloheptyl-N-methylsulfonyl-4-(2-quinolinyl-methoxy)-phenyl-acetamide BAYER AG (DE) 1994-04-27 EP disclosed
EP-0593976-A1 Crystalline (R)-(-)-2-cycloheptyl-N-methylsulfonyl-4-(2-quinolinyl-methoxy)-phenyl-acetamide BAYER AG (DE) 1994-04-27 EP disclosed