SCHEMBL6441833

SCHEMBL6441833

COC(=O)COc1ccc2c(c1)C[C@H](NC[C@H](O)c1cccc(Cl)c1)CC2

nearest known ligand 0.84

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 15/20 0.83
ADRB1 P08588 4/20 0.83

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9006798 1.00 ADRB3 (0.83) ADRB3ADRB1
Hydrochloric Acid SCHEMBL9317518 0.99 ADRB3 (0.82) ADRB3ADRB1
Amibegron SCHEMBL2052478 0.92 ADRB3 (0.91) ADRB3ADRB1
Amibegron SCHEMBL6931932 0.92 ADRB3 (0.91) ADRB3ADRB1
Amibegron SCHEMBL29373533 0.92 ADRB3 (0.91) ADRB3ADRB1
Amibegron SCHEMBL9006793 0.92 ADRB3 (0.91) ADRB3ADRB1
Amibegron SCHEMBL5200899 0.92 ADRB3 (0.91) ADRB3ADRB1
Amibegron SCHEMBL3898164 0.92 ADRB3 (0.91) ADRB3ADRB1
Amibegron SCHEMBL8765764 0.92 ADRB3 (0.91) ADRB3ADRB1
Amibegron SCHEMBL3824162 0.92 ADRB3 (0.91) ADRB3ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966276-B1 USE OF BETA-3 ADRENERGIC RECEPTOR AGONISTS FOR PREPARING WOUND-HEALING PHARMACEUTICALS SANOFI SYNTHELABO (FR) 2003-12-10 EP claimed
EP-0403360-B1 Use of phenylethanolamines for the preparation of a medicament for treating ophthalmologic disorders SANOFI SA (FR) 1996-10-16 EP claimed
EP-0303546-B1 O-alkylation process for N-(hydroxy)aralkyl phenyl ethanol amines SANOFI SA (FR) 1994-12-28 EP claimed
EP-0403360-A2 Use of phenylethanolamines for the preparation of a medicament for treating ophthalmologic disorders SANOFI (FR) 1990-12-19 EP claimed
US-4927955-A Process for the O-alkylation of N-(hydroxy)aralkylphenylethanolamines SANOFI (FR) 1990-05-22 US claimed
EP-0303546-A2 O-alkylation process for N-(hydroxy)aralkyl phenyl ethanol amines SANOFI (FR) 1989-02-15 EP claimed
US-20050026986-A1 Use of central cannabinoid receptor antagonists for the preparation of drugs SANOFI-AVENTIS (FR) 2005-02-03 US disclosed
EP-0966276-B1 USE OF BETA-3 ADRENERGIC RECEPTOR AGONISTS FOR PREPARING WOUND-HEALING PHARMACEUTICALS SANOFI SYNTHELABO (FR) 2003-12-10 EP disclosed
US-20020128302-A1 Use of central cannabinoid receptor antagonists for the preparation of drugs MARUANI JEANNE (FR) 2002-09-12 US disclosed
US-6344474-B1 Use of central cannabinoid receptor antagonists for regulating appetence SANOFI-SYNTHELABO (FR) 2002-02-05 US disclosed
EP-0969835-A1 USE OF CENTRAL CANNABINOID RECEPTOR ANTAGONISTS FOR REGULATING APPETENCE SANOFI-SYNTHELABO (FR) 2000-01-12 EP disclosed
EP-0966276-A1 USE OF AGONISTS OF ADRENERGIC BETA-3 RECEPTORS FOR PREPARING WOUND-HEALING MEDICINES SANOFI-SYNTHELABO (FR) 1999-12-29 EP disclosed
WO-1998032441-A1 USE OF CENTRAL CANNABINOID RECEPTOR ANTAGONISTS FOR REGULATING APPETENCE SANOFI-SYNTHELABO (FR) 1998-07-30 WO disclosed
EP-0303546-B1 O-alkylation process for N-(hydroxy)aralkyl phenyl ethanol amines SANOFI SA (FR) 1994-12-28 EP disclosed
US-5347037-A (RR) and (RS stereoisomers of N-(7-ethoxycarbonylmethoxy-1,2,3,-tetrahydronaphth-2-yl)-2-(3-chlorophenyl)-2-hydroxyethanamine and their pharmaceutically acceptable salts SANOFI (FR) 1994-09-13 US disclosed
US-5236951-A Administering a phenylethanolamine derivative SANOFI (FR) 1993-08-17 US disclosed
US-5041606-A Process for the O-alkylation of N-(hydroxy)aralkylphenylethanolamines SANOFI 1991-08-20 US disclosed
EP-0403360-A2 Use of phenylethanolamines for the preparation of a medicament for treating ophthalmologic disorders SANOFI (FR) 1990-12-19 EP disclosed
US-4927955-A Process for the O-alkylation of N-(hydroxy)aralkylphenylethanolamines SANOFI (FR) 1990-05-22 US disclosed
EP-0303546-A2 O-alkylation process for N-(hydroxy)aralkyl phenyl ethanol amines SANOFI (FR) 1989-02-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050026986-A1 Use of central cannabinoid receptor antagonists for the preparation of drugs CNR1, CNR2, ADRB3 ADRB3 3/4885ADRB1 4/4885
US-20020128302-A1 Use of central cannabinoid receptor antagonists for the preparation of drugs CNR1, CNR2, GPR119 ADRB3 4/4885ADRB1 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.