SCHEMBL6442855

SCHEMBL6442855

CS(=O)(=O)c1ccc(-c2[nH]nc(C(=O)CCCO)c2-c2ccc(F)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 2/20 0.47
PTGS2 P35354 15/20 0.45
CDC25B P30305 2/20 0.44
PTGS1 P23219 2/20 0.42
MAPK13 O15264 1/20 0.41
RAF1 P04049 1/20 0.41
MAPK9 P45984 1/20 0.41
MAPK12 P53778 1/20 0.41
MAPK11 Q15759 1/20 0.41
MAPK14 Q16539 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6438854 0.90 PTGS2 (0.43) ESR2PTGS2CDC25BPTGS1
SCHEMBL6444404 0.90 PTGS2 (0.44) ESR2PTGS2CDC25BPTGS1
SCHEMBL6438518 0.89 PTGS2 (0.44) ESR2PTGS2CDC25B
SCHEMBL5674799 0.89 PTGS2 (0.44) PTGS2CDC25BPTGS1
SCHEMBL3865448 0.86 PTGS2 (0.40) ESR2PTGS2CDC25BMAPK9
SCHEMBL6440170 0.86 ESR2 (0.49) ESR2PTGS2CDC25BPTGS1
SCHEMBL6470454 0.81 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL3865463 0.76 ESR2 (0.49) ESR2PTGS2CDC25BPTGS1
SCHEMBL7539198 0.76 PTGS2 (0.56) PTGS2PTGS1
SCHEMBL6620090 0.76 PTGS2 (0.56) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP claimed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP claimed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO claimed