SCHEMBL6440170

SCHEMBL6440170

CS(=O)(=O)c1ccc(-c2[nH]nc(C(=O)CCCO[N+](=O)[O-])c2-c2ccc(F)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 2/20 0.49
PTGS2 P35354 10/20 0.45
PTGS1 P23219 2/20 0.45
CDC25B P30305 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3865463 0.91 ESR2 (0.49) ESR2PTGS2PTGS1CDC25B
SCHEMBL6438007 0.90 PTGS2 (0.45) ESR2PTGS2PTGS1CDC25B
SCHEMBL6439987 0.90 PTGS2 (0.45) ESR2PTGS2PTGS1CDC25B
SCHEMBL6442807 0.90 PTGS2 (0.43) ESR2PTGS2PTGS1
SCHEMBL3865578 0.88 PTGS2 (0.43) ESR2PTGS2PTGS1CDC25B
SCHEMBL6442855 0.86 ESR2 (0.47) ESR2PTGS2PTGS1CDC25B
SCHEMBL6438240 0.80 PTGS2 (0.48) ESR2PTGS2PTGS1
SCHEMBL5150520 0.79 ESR2 (0.47) ESR2PTGS2PTGS1
SCHEMBL6470454 0.78 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL6444404 0.77 PTGS2 (0.44) ESR2PTGS2PTGS1CDC25B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP disclosed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP disclosed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed