SCHEMBL6442958

SCHEMBL6442958

COCc1cc(NC(C)CCCN2C(=O)c3ccccc3C2=O)c2ncccc2c1Oc1ccc(Cl)c(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 7/20 0.44
MAOB P27338 7/20 0.44
KDM4E B2RXH2 3/20 0.44
MAPT P10636 3/20 0.44
NSD2 O96028 1/20 0.44
HSP90AA1 P07900 2/20 0.41
HSP90AB1 P08238 2/20 0.41
CASP7 P55210 2/20 0.40
CASP6 P55212 2/20 0.40
PABPC1 P11940 1/20 0.40
IDO1 P14902 1/20 0.36
CYP1A2 P05177 2/20 0.36
CASP1 P29466 2/20 0.36
LMNA P02545 2/20 0.36
ABCB11 O95342 1/20 0.36
ESR1 P03372 1/20 0.36
PGR P06401 1/20 0.36
ADRB2 P07550 1/20 0.36
CHRM2 P08172 1/20 0.36
ADRB1 P08588 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11545426 0.83 KDM4E (0.59) MAOAMAOBKDM4EMAPTNSD2
SCHEMBL14534512 0.80 MAOA (0.60) MAOAMAOBKDM4EMAPTNSD2
SCHEMBL5493085 0.79 MAOA (0.72) MAOAMAOBKDM4EMAPTNSD2
SCHEMBL6442964 0.78 MAOA (0.50) MAOAMAOBKDM4EMAPTNSD2
SCHEMBL10949994 0.76 HSP90AA1 (0.56) MAOAMAOBKDM4EMAPTNSD2
SCHEMBL10944231 0.76 HSP90AA1 (0.58) MAOAMAOBKDM4EMAPTNSD2
SCHEMBL10944622 0.75 HSP90AA1 (0.56) MAOAMAOBKDM4EMAPTNSD2
SCHEMBL4726838 0.74 HSP90AA1 (0.52) MAOAMAOBKDM4EMAPTNSD2
SCHEMBL10942299 0.73 HSP90AA1 (0.54) MAOAMAOBKDM4EMAPTNSD2
SCHEMBL10941487 0.73 HSP90AA1 (0.54) MAOAMAOBKDM4EMAPTNSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0907363-A4 8-AMINOQUINOLINES UNIV MISSISSIPPI (US) 2005-04-06 EP disclosed
EP-0907363-A1 8-AMINOQUINOLINES THE UNIVERSITY OF MISSISSIPPI (US) 1999-04-14 EP disclosed
WO-1997036590-A1 8-AMINOQUINOLINES THE UNIVERSITY OF MISSISSIPPI (US) 1997-10-09 WO disclosed