SCHEMBL6443162

SCHEMBL6443162

CCCCCCOC(=O)NCC(C(=O)NCC#N)S(C)(=O)=O

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
LMNA P02545 1/20 0.48
ACHE P22303 12/20 0.44
EPHX1 P07099 1/20 0.42
CTSS P25774 2/20 0.40
CTSL P07711 1/20 0.40
EPHX2 P34913 2/20 0.39
CTSK P43235 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6447728 0.95 NPC1 (0.44) NPC1RAB9ASMN1; SMN2LMNAACHE
SCHEMBL6446210 0.90 ACHE (0.45) NPC1RAB9ASMN1; SMN2LMNAACHE
SCHEMBL6443436 0.84 ACHE (0.40) NPC1RAB9ASMN1; SMN2LMNAACHE
SCHEMBL6822996 0.82 CTSS (0.38) CTSSCTSLCTSK
SCHEMBL6447218 0.80 CTSS (0.40) CTSSCTSLCTSK
SCHEMBL6443215 0.80 NPC1 (0.49) NPC1RAB9ASMN1; SMN2LMNAACHE
SCHEMBL6443744 0.80 CTSS (0.42) SMN1; SMN2LMNACTSSCTSLCTSK
SCHEMBL6443769 0.78 NPC1 (0.65) NPC1RAB9ASMN1; SMN2LMNACTSS
SCHEMBL6020800 0.77 CTSS (0.49) NPC1RAB9ASMN1; SMN2ACHEEPHX1
SCHEMBL6442459 0.76 SMN1; SMN2 (0.54) NPC1RAB9ASMN1; SMN2LMNAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed