SCHEMBL6445534

SCHEMBL6445534

Cc1ccc(S(=O)(=O)N2CCc3ccccc3C2)cc1C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.78
KMT2A Q03164 4/20 0.78
SMN1; SMN2 Q16637 2/20 0.66
CYP3A4 P08684 1/20 0.66
CYP2C19 P33261 1/20 0.66
NPSR1 Q6W5P4 1/20 0.66
RAB9A P51151 1/20 0.61
POLB P06746 1/20 0.61
MAPK1 P28482 1/20 0.60
AKR1C3 P42330 5/20 0.59
AKR1C1 Q04828 1/20 0.59
ALDH1A1 P00352 3/20 0.57
PKM P14618 1/20 0.57
KDM4E B2RXH2 1/20 0.57
HPGD P15428 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13302259 0.84 KMT2A (0.77) MEN1KMT2ASMN1; SMN2CYP3A4CYP2C19
SCHEMBL8589869 0.81 MEN1 (0.68) MEN1KMT2ASMN1; SMN2CYP3A4CYP2C19
SCHEMBL693455 0.80 KMT2A (1.00) MEN1KMT2ASMN1; SMN2CYP3A4CYP2C19
SCHEMBL6429647 0.80 CYP3A4 (1.00) MEN1KMT2ASMN1; SMN2CYP3A4CYP2C19
SCHEMBL12793350 0.78 KMT2A (0.77) MEN1KMT2ASMN1; SMN2CYP3A4CYP2C19
SCHEMBL21067983 0.78 KMT2A (0.82) MEN1KMT2ASMN1; SMN2CYP3A4CYP2C19
SCHEMBL5915341 0.78 KMT2A (0.77) MEN1KMT2ASMN1; SMN2CYP3A4CYP2C19
SCHEMBL29941108 0.78 KMT2A (0.82) MEN1KMT2ASMN1; SMN2CYP3A4CYP2C19
SCHEMBL20389408 0.78 KMT2A (0.77) MEN1KMT2ASMN1; SMN2CYP3A4CYP2C19
SCHEMBL25442198 0.77 MEN1 (0.70) MEN1KMT2ASMN1; SMN2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP claimed
JP-2002512625-A 2002-04-23 JP claimed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP claimed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO claimed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed