SCHEMBL6446129

SCHEMBL6446129

CC(C)CCNC(=O)/C=C\C(CCc1ccccc1)O[Si](C)(C)C(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.46
PKM P14618 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 5/20 0.41
TAAR1 Q96RJ0 2/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HTT P42858 1/20 0.40
KCNA5 P22460 1/20 0.40
MMP1 P03956 1/20 0.40
POLB P06746 1/20 0.40
MMP2 P08253 1/20 0.40
MMP9 P14780 1/20 0.40
RECQL P46063 1/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
ANPEP P15144 2/20 0.39
RNPEP Q9H4A4 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446132 1.00 LMNA (0.46) LMNAPKML3MBTL1ALDH1A1TAAR1
SCHEMBL6446733 0.84 HCAR2 (0.40) ALDH1A1TAAR1HPGDSMN1; SMN2HTT
SCHEMBL6450631 0.84 HCAR2 (0.40) ALDH1A1TAAR1HPGDSMN1; SMN2HTT
SCHEMBL6446730 0.84 HCAR2 (0.40) ALDH1A1TAAR1HPGDSMN1; SMN2HTT
SCHEMBL7268895 0.78 LMNA (0.58) LMNAPKML3MBTL1ALDH1A1TAAR1
SCHEMBL7268887 0.78 LMNA (0.58) LMNAPKML3MBTL1ALDH1A1TAAR1
SCHEMBL4494121 0.78 PRSS1 (0.34) ALDH1A1HPGDSMN1; SMN2HTTCYP2C9
SCHEMBL7552716 0.78 PRSS1 (0.34) ALDH1A1HPGDSMN1; SMN2HTTCYP2C9
SCHEMBL4494128 0.78 PRSS1 (0.34) ALDH1A1HPGDSMN1; SMN2HTTCYP2C9
SCHEMBL7552725 0.78 PRSS1 (0.34) ALDH1A1HPGDSMN1; SMN2HTTCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-B1 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LAB (US) 2005-08-17 EP disclosed
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed