SCHEMBL6446733

SCHEMBL6446733

CC(C)(C)[Si](C)(C)OC(C=CC(=O)O)CCc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.40
SLC15A1 P46059 1/20 0.38
PRSS1 P07477 2/20 0.38
CTSG P08311 2/20 0.38
CTRB1 P17538 2/20 0.38
CMA1 P23946 2/20 0.38
CTSL P07711 1/20 0.38
ALDH1A1 P00352 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
MAPK1 P28482 1/20 0.37
CYP2C19 P33261 1/20 0.37
TAAR1 Q96RJ0 2/20 0.37
TSHR P16473 1/20 0.37
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6450631 1.00 HCAR2 (0.40) HCAR2SLC15A1PRSS1CTSGCTRB1
SCHEMBL6446730 1.00 HCAR2 (0.40) HCAR2SLC15A1PRSS1CTSGCTRB1
SCHEMBL7552716 0.85 PRSS1 (0.34) PRSS1CTSGCTRB1CMA1ALDH1A1
SCHEMBL4494128 0.85 PRSS1 (0.34) PRSS1CTSGCTRB1CMA1ALDH1A1
SCHEMBL7552725 0.85 PRSS1 (0.34) PRSS1CTSGCTRB1CMA1ALDH1A1
SCHEMBL4494121 0.85 PRSS1 (0.34) PRSS1CTSGCTRB1CMA1ALDH1A1
SCHEMBL6446129 0.84 LMNA (0.46) ALDH1A1CYP1A2CYP3A4CYP2C9MAPK1
SCHEMBL6446132 0.84 LMNA (0.46) ALDH1A1CYP1A2CYP3A4CYP2C9MAPK1
SCHEMBL12549853 0.84 PRSS1 (0.33) PRSS1CTSGCTRB1CMA1
SCHEMBL17429760 0.83 PRSS1 (0.32) PRSS1CTSGCTRB1CMA1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-B1 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LAB (US) 2005-08-17 EP disclosed
EP-0402646-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 1998-07-22 EP disclosed
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed