SCHEMBL6446459

SCHEMBL6446459

CC(C)C(NC(=O)OCc1ccncc1)C(=O)Oc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.51
MMP13 P45452 2/20 0.45
ALDH1A1 P00352 2/20 0.43
GAA P10253 2/20 0.43
MAPT P10636 2/20 0.43
ELANE P08246 1/20 0.43
SLC2A1 P11166 1/20 0.42
MGLL Q99685 1/20 0.41
POLB P06746 1/20 0.41
ADAMTS4 O75173 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446463 1.00 HTR2A (0.51) HTR2AMMP13ALDH1A1GAAMAPT
SCHEMBL7333604 0.89 HTR2A (0.53) HTR2AELANE
SCHEMBL7328473 0.89 HTR2A (0.53) HTR2AELANE
SCHEMBL6447457 0.88 MAPT (0.48) HTR2AALDH1A1GAAMAPTELANE
SCHEMBL6447461 0.88 MAPT (0.48) HTR2AALDH1A1GAAMAPTELANE
SCHEMBL4679034 0.82 KMT2A (0.48) HTR2AALDH1A1GAAMAPTELANE
SCHEMBL4679037 0.82 KMT2A (0.48) HTR2AALDH1A1GAAMAPTELANE
SCHEMBL7308656 0.82 CYP3A4 (0.44) HTR2AALDH1A1GAAMAPTMGLL
SCHEMBL7308651 0.82 CYP3A4 (0.44) HTR2AALDH1A1GAAMAPTMGLL
SCHEMBL11771667 0.80 CTSL (0.55) HTR2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-B1 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LAB (US) 2005-08-17 EP disclosed
EP-0402646-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 1998-07-22 EP disclosed
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed