SCHEMBL7333604

SCHEMBL7333604

CC(C)C(NC(=O)OCc1ccccc1)C(=O)Oc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.53
ELANE P08246 3/20 0.50
CTSL P07711 4/20 0.49
CTSB P07858 1/20 0.49
CTSS P25774 1/20 0.49
CTSK P43235 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
PRTN3 P24158 1/20 0.47
CA2 P00918 1/20 0.47
CA5A P35218 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7328473 1.00 HTR2A (0.53) HTR2AELANECTSLCTSBCTSS
SCHEMBL7278888 0.90 CTSL (0.55) HTR2ACTSLCTSBCTSSCTSK
SCHEMBL7278892 0.90 CTSL (0.55) HTR2ACTSLCTSBCTSSCTSK
SCHEMBL11771667 0.90 CTSL (0.55) HTR2ACTSLCTSBCTSSCTSK
SCHEMBL29838911 0.90 HTR2A (0.55) HTR2AELANECTSLCTSBCTSS
SCHEMBL8432555 0.90 CTSB (0.53) CTSLCTSBCTSSCTSKMEN1
SCHEMBL1801469 0.90 HTR2A (0.56) HTR2ACTSLCTSBCTSSCTSK
SCHEMBL10794620 0.90 HTR2A (0.56) HTR2ACTSLCTSBCTSSCTSK
SCHEMBL8432553 0.90 CTSB (0.53) CTSLCTSBCTSSCTSKMEN1
SCHEMBL6446459 0.89 HTR2A (0.51) HTR2AELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3038553-A None JP disclosed
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed
JP-H0338553-A ASYMMETRICALLY REACTIVE INORGANIC OXIDE POWDER CARRYING AMINO ACID OSAKA ORGANIC CHEM IND LTD 1991-02-19 JP disclosed