SCHEMBL6446462

SCHEMBL6446462

CC(C)[C@H](NC(=O)OCc1cccnc1)C(=O)N[C@@H](Cc1ccccc1)[C@@H](O)[C@@H](O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSD P07339 3/20 0.56
BACE1 P56817 5/20 0.53
KLK5 Q9Y337 1/20 0.52
CYP3A4 P08684 1/20 0.49
PSEN1 P49768 2/20 0.49
PSEN2 P49810 2/20 0.49
APH1B Q8WW43 2/20 0.49
NCSTN Q92542 2/20 0.49
APH1A Q96BI3 2/20 0.49
PSENEN Q9NZ42 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6448343 0.93 CTSD (0.63) CTSDCYP3A4
SCHEMBL6449478 0.93 CTSD (0.63) CTSDCYP3A4
SCHEMBL6446319 0.93 CTSD (0.63) CTSDCYP3A4
SCHEMBL7430958 0.91 BACE1 (0.61) CTSDBACE1KLK5
SCHEMBL6449655 0.91 CTSD (0.66) CTSDBACE1KLK5PSEN1PSEN2
SCHEMBL7268971 0.91 CTSD (0.63) CTSDCYP3A4
SCHEMBL6444641 0.90 CTSD (0.51) CTSDBACE1KLK5CYP3A4
SCHEMBL7275770 0.90 CTSD (0.65) CTSDCYP3A4
SCHEMBL15095216 0.90 CTSD (0.67) CTSDBACE1KLK5PSEN1PSEN2
SCHEMBL6447745 0.89 CTSD (0.66) CTSDBACE1KLK5PSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-B1 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LAB (US) 2005-08-17 EP disclosed
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed