SCHEMBL7430958

SCHEMBL7430958

CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)NC(Cc1ccncc1)C(O)C(O)C(Cc1ccncc1)NC(=O)OC(C)(C)C

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 11/20 0.61
CTSD P07339 3/20 0.60
KLK5 Q9Y337 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6449655 0.94 CTSD (0.66) BACE1CTSDKLK5
SCHEMBL15095216 0.93 CTSD (0.67) BACE1CTSDKLK5
SCHEMBL6447745 0.93 CTSD (0.66) BACE1CTSDKLK5
SCHEMBL6448985 0.92 CTSD (0.68) BACE1CTSD
SCHEMBL6454320 0.92 CTSD (0.68) BACE1CTSD
SCHEMBL7270278 0.92 CTSD (0.67) BACE1CTSDKLK5
SCHEMBL6446462 0.91 CTSD (0.56) BACE1CTSDKLK5
SCHEMBL6449617 0.91 CTSD (0.68) BACE1CTSD
SCHEMBL7268574 0.91 CTSD (0.68) BACE1CTSD
SCHEMBL7443260 0.88 CTSD (0.59) BACE1CTSDKLK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018866-A2 1,4-DIAMINO-2,3-DIHYDROXYBUTANES THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1991-12-12 WO claimed
EP-0665215-A1 1,4-Diamino-2,3-dihydroxybutanes THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-08-02 EP disclosed