SCHEMBL6447189

SCHEMBL6447189

CSC(CNC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)NCC#N

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.49
CASP3 P42574 3/20 0.43
EPHX2 P34913 1/20 0.42
CTSS P25774 4/20 0.40
CTSL P07711 3/20 0.40
CTSB P07858 2/20 0.40
CTSK P43235 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6443477 0.85 KMT2A (0.49) KMT2ACASP3EPHX2CTSSCTSL
SCHEMBL6446919 0.84 CASP3 (0.49) KMT2ACASP3EPHX2CTSSCTSL
SCHEMBL6019629 0.82 CTSS (0.51) KMT2ACASP3CTSSCTSLCTSB
SCHEMBL6443951 0.81 KMT2A (0.46) KMT2ACASP3EPHX2CTSSCTSL
SCHEMBL6019554 0.77 CTSS (0.69) CTSSCTSLCTSBCTSK
SCHEMBL12461580 0.77 KMT2A (0.57) KMT2ACASP3EPHX2
SCHEMBL31670673 0.77 KMT2A (0.57) KMT2ACASP3EPHX2
SCHEMBL60494 0.77 KMT2A (0.57) KMT2ACASP3EPHX2
SCHEMBL15727228 0.77 KMT2A (0.57) KMT2ACASP3EPHX2
SCHEMBL3740743 0.77 KMT2A (0.57) KMT2ACASP3EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed