SCHEMBL644763

SCHEMBL644763

C=CCOC(=O)NC(CC(=O)O)C(O)COC(=O)c1cccc(O)c1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.44
ADRB1 P08588 2/20 0.44
ADRB3 P13945 2/20 0.44
CASP1 P29466 16/20 0.43
ALDH1A1 P00352 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1410176 0.87 ADRB2 (0.47) ADRB2ADRB1ADRB3CASP1ALDH1A1
SCHEMBL646188 0.81 CASP1 (0.44) CASP1
SCHEMBL646998 0.81 CASP1 (0.53) ADRB2ADRB1ADRB3CASP1ALDH1A1
SCHEMBL10201585 0.76 ADRB2 (0.46) ADRB2ADRB1ADRB3CASP1ALDH1A1
SCHEMBL647269 0.76 CASP1 (0.48) ADRB2ADRB1ADRB3CASP1
SCHEMBL2787842 0.76 CYP3A4 (0.54) ADRB2ADRB1ADRB3ALDH1A1NPC1
SCHEMBL10918370 0.74 CYP3A4 (0.53) ADRB2ADRB1ADRB3ALDH1A1NPC1
SCHEMBL645196 0.72 CASP1 (0.45) CASP1
Benzene SCHEMBL29140663 0.69 CYP3A4 (0.59) ADRB2ADRB1ADRB3ALDH1A1NPC1
SCHEMBL311041 0.69 KLK5 (0.36) ADRB2ADRB1ADRB3CASP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119631-B2 Inhibitors of interleukin-1β converting enzyme VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-02-21 US disclosed