SCHEMBL6448199

SCHEMBL6448199

COC(=O)[C@@H](NC(=O)OCCN1CCOCC1)C(C)C

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.45
ALDH1A1 P00352 5/20 0.44
KDM4E B2RXH2 2/20 0.44
HPGD P15428 2/20 0.44
ATM Q13315 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
ACACB O00763 1/20 0.42
TSHR P16473 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
LMNA P02545 2/20 0.40
KMT2A Q03164 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6448194 1.00 TDP1 (0.45) TDP1ALDH1A1KDM4EHPGDATM
SCHEMBL6444915 0.89 ALDH1A1 (0.47) TDP1ALDH1A1KDM4EHPGDATM
SCHEMBL6444920 0.89 ALDH1A1 (0.47) TDP1ALDH1A1KDM4EHPGDATM
SCHEMBL6446180 0.88 ALDH1A1 (0.46) TDP1ALDH1A1KDM4EHPGDATM
SCHEMBL6446187 0.88 ALDH1A1 (0.46) TDP1ALDH1A1KDM4EHPGDATM
SCHEMBL7279077 0.87 TSHR (0.41) ATMACACBTSHRKMT2A
SCHEMBL7279082 0.87 TSHR (0.41) ATMACACBTSHRKMT2A
Lithium Ion SCHEMBL6446186 0.86 ALDH1A1 (0.42) TDP1ALDH1A1KDM4EHPGDATM
SCHEMBL25669794 0.84 HRH3 (0.50) TDP1ALDH1A1KDM4EHPGDATM
SCHEMBL18427273 0.79 ALDH1A1 (0.54) TDP1ALDH1A1KDM4EHPGDATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-B1 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LAB (US) 2005-08-17 EP disclosed
EP-0402646-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 1998-07-22 EP disclosed
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed