SCHEMBL644937

SCHEMBL644937

O=C1c2ccccc2C(=O)N1CC=CCCl

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.51
CA12 O43570 1/20 0.44
CA9 Q16790 1/20 0.44
GLS O94925 1/20 0.44
ALDH1A1 P00352 2/20 0.42
ALDH3A1 P30838 1/20 0.41
RCE1 Q9Y256 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2319856 1.00 CASP3 (0.51) CASP3CA12CA9GLSALDH1A1
SCHEMBL643984 1.00 CASP3 (0.51) CASP3CA12CA9GLSALDH1A1
SCHEMBL4476083 0.90 CASP3 (0.60) CASP3CA12CA9GLSALDH1A1
SCHEMBL8950475 0.90 CASP3 (0.60) CASP3CA12CA9GLSALDH1A1
SCHEMBL4468251 0.90 CASP3 (0.60) CASP3CA12CA9GLSALDH1A1
SCHEMBL21901972 0.82 CASP3 (0.53) CASP3CA12CA9GLSALDH1A1
SCHEMBL25302148 0.81 CASP3 (0.51) CASP3CA12CA9GLSALDH1A1
SCHEMBL9761279 0.81 CASP3 (0.51) CASP3CA12CA9GLSALDH1A1
SCHEMBL23077378 0.81 CASP3 (0.51) CASP3CA12CA9GLSALDH1A1
SCHEMBL12439955 0.81 CASP3 (0.51) CASP3CA12CA9GLSALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 79 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317416-A2 2-AMINO-2-ALKYL-4 HEXENOIC AND HEXYNOIC ACID DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS Pharmacia Corporation (US) 2003-06-11 EP claimed
WO-2002022559-A2 2-AMINO-2-ALKYL-4 HEXENOIC AND HEXYNOIC ACID DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS PHARMACIA CORPORATION (US) 2002-03-21 WO claimed
JP-3227962-A None JP disclosed
US-12582645-B2 Chemokine CXCR4 receptor modulators and uses related thereto EMORY UNIVERSITY (US) 2026-03-24 US disclosed
US-20240316034-A1 Chemokine CXCR4 Receptor Modulators and Uses Related Thereto UNIV EMORY (US) 2024-09-26 US disclosed
US-20230112832-A1 Chemokine CXCR4 Receptor Modulators and Uses Related Thereto UNIV EMORY (US) 2023-04-13 US disclosed
US-11497744-B2 Chemokine CXCR4 receptor modulators and uses related thereto EMORY UNIVERSITY (US) 2022-11-15 US disclosed
US-20200054623-A1 Chemokine CXCR4 Receptor Modulators and Uses Related Thereto EMORY UNIVERSITY 2020-02-20 US disclosed
CN-110545814-A Chemokine CXCR4 receptor modulators and uses related thereto UNIV EMORY 2019-12-06 CN disclosed
WO-2018156595-A1 CHEMOKINE CXCR4 RECEPTOR MODULATORS AND USES RELATED THERETO EMORY UNIVERSITY (US) 2018-08-30 WO disclosed
EP-2354136-B1 NOVEL DOPAMINE D3 RECEPTOR LIGANDS AND PREPARATION AND MEDICAL USES OF THE SAME INST PHARM & TOXICOLOGY AMMS (CN) 2016-02-24 EP disclosed
EP-0641789-B1 BENZOTHIADIAZINE DERIVATIVE TAIHO PHARMACEUTICAL CO LTD (JP) 1997-12-03 EP disclosed
US-5401739-A Benzothiadiazine derivatives TAIHO PHARMACEUTICAL CO. LTD. (JP) 1995-03-28 US disclosed
EP-0641789-A1 BENZOTHIADIAZINE DERIVATIVE TAIHO PHARMACEUTICAL COMPANY LIMITED (JP) 1995-03-08 EP disclosed
EP-0625978-A1 PIPERAZINE AND PIPERIDINE DERIVATIVES, AND THEIR USE AS ANTIPSYCHOTICS THE WELLCOME FOUNDATION LIMITED (GB) 1994-11-30 EP disclosed
WO-1993016073-A1 PIPERAZINE AND PIPERIDINE DERIVATIVES, AND THEIR USE AS ANTIPSYCHOTICS THE WELLCOME FOUNDATION LIMITED (GB) 1993-08-19 WO disclosed
JP-H03227962-A PRODUCTION OF 4-AMINO-CIS-2-BUTEN-1-OL IKEDA MOHANDOU:KK 1991-10-08 JP disclosed
US-4568687-A THROMBOXANE SYNTHETASE TNZYME INHIBITORS; HYPOTENSIVE AGENTS, CARDIOTONIC AGENTS AMERICAN CYANAMID COMPANY (US) 1986-02-04 US disclosed
US-4489089-A INHIBITION OF THE ENZYME THROMBOXANE SYNTHETASE AMERICAN CYANAMID COMPANY (US) 1984-12-18 US disclosed
EP-0117462-A2 N-(2-4-(1H-imidazol-1-yl)alkyl)arylamides AMERICAN CYANAMID COMPANY (US) 1984-09-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200054623-A1 Chemokine CXCR4 Receptor Modulators and Uses Related Thereto CXCR4, CXCL12, CXCR1 CASP3 2722/4885CA12 3520/4885CA9 3149/4885
US-20240316034-A1 Chemokine CXCR4 Receptor Modulators and Uses Related Thereto CXCR4, CXCL12, CXCR1 CASP3 2722/4885CA12 3520/4885CA9 3149/4885
US-11497744-B2 Chemokine CXCR4 receptor modulators and uses related thereto CXCR4, CXCL12, CXCR1 CASP3 2722/4885CA12 3520/4885CA9 3149/4885
US-20230112832-A1 Chemokine CXCR4 Receptor Modulators and Uses Related Thereto CXCR4, CXCL12, CXCR1 CASP3 2722/4885CA12 3520/4885CA9 3149/4885
US-12582645-B2 Chemokine CXCR4 receptor modulators and uses related thereto CXCR4, CXCR2, CXCR1 CASP3 2144/4885CA12 2293/4885CA9 3659/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.