SCHEMBL6449536

SCHEMBL6449536

CCCc1c(OC)cc(/C=C/c2c(F)cccc2F)cc1OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP1B1 Q16678 1/20 0.44
NFE2L2 Q16236 3/20 0.44
TUBB1 Q9H4B7 7/20 0.43
KRAS P01116 2/20 0.43
PTGS1 P23219 2/20 0.42
KCNH2 Q12809 4/20 0.41
MAT2A P31153 1/20 0.41
ALOX5 P09917 2/20 0.41
PTGS2 P35354 1/20 0.41
TUBB4A P04350 3/20 0.40
TUBB P07437 3/20 0.40
TUBA3C P0DPH7 3/20 0.40
TUBA1B P68363 3/20 0.40
TUBA4A P68366 3/20 0.40
TUBB4B P68371 3/20 0.40
TUBB3 Q13509 3/20 0.40
TUBB2A Q13885 3/20 0.40
TUBB8 Q3ZCM7 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL918372 1.00 CYP1A1 (0.44) CYP1A1CYP1A2CYP1B1NFE2L2TUBB1
SCHEMBL6450850 0.87 TUBB1 (0.41) CYP1A1CYP1A2CYP1B1NFE2L2TUBB1
SCHEMBL919181 0.87 TUBB1 (0.41) CYP1A1CYP1A2CYP1B1NFE2L2TUBB1
SCHEMBL917823 0.84 NFE2L2 (0.56) CYP1A1CYP1A2CYP1B1NFE2L2TUBB1
SCHEMBL6448424 0.84 TUBB1 (0.41) CYP1A1CYP1A2CYP1B1NFE2L2TUBB1
SCHEMBL917832 0.84 TUBB1 (0.41) CYP1A1CYP1A2CYP1B1NFE2L2TUBB1
SCHEMBL919199 0.83 NFE2L2 (0.64) NFE2L2TUBB1PTGS1ALOX5PTGS2
SCHEMBL6448352 0.81 CYP1A1 (0.45) CYP1A1CYP1A2CYP1B1NFE2L2TUBB1
SCHEMBL918373 0.81 NFE2L2 (0.61) NFE2L2TUBB1PTGS1TUBB4ATUBB
SCHEMBL6453082 0.81 NFE2L2 (0.61) NFE2L2TUBB1PTGS1TUBB4ATUBB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1554236-A1 NOVEL BIOACTIVE DIPHENYL ETHENE COMPOUNDS AND THEIR THERAPEUTIC APPLICATIONS Welichem Biotech Inc. (CA) 2005-07-20 EP disclosed
WO-2004031117-A1 NOVEL BIOACTIVE DIPHENYL ETHENE COMPOUNDS AND THEIR THERAPEUTIC APPLICATIONS WELICHEM BIOTECH INC. (CA) 2004-04-15 WO disclosed