SCHEMBL6450281

SCHEMBL6450281

COc1cc(CC#Cc2cc3c(=O)[nH]cc(Cc4ccc(S(C)(=O)=O)cc4)c3s2)ccn1

nearest known ligand 0.31

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PLA2G7 Q13093 1/20 0.31
LOX P28300 1/20 0.31
LOXL2 Q9Y4K0 1/20 0.31
CDK4 P11802 1/20 0.30
CCND1 P24385 1/20 0.30
CDK2 P24941 1/20 0.30
DAO P14920 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6237217 0.77 MMP13 (0.36)
SCHEMBL6477603 0.76 LOX (0.31) LOXLOXL2
SCHEMBL6234429 0.76 LOX (0.31) LOXLOXL2
SCHEMBL6232535 0.74 MMP13 (0.36) LOXLOXL2
SCHEMBL6258139 0.73 TRPA1 (0.39)
SCHEMBL6258372 0.70 FFAR1 (0.34) LOXLOXL2
SCHEMBL6296263 0.64 MMP13 (0.60)
SCHEMBL6296207 0.64 MMP13 (0.53)
SCHEMBL6231728 0.64 MMP13 (0.49)
SCHEMBL6487927 0.63 CYP3A4 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534274-A1 COMBINATION OF AN ALLOSTERIC ALKYNE INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB Warner-Lambert Company LLC (US) 2005-06-01 EP disclosed
WO-2004006914-A1 COMBINATION OF AN ALLOSTERIC ALKYNE INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed