SCHEMBL6450666

SCHEMBL6450666

CCCCCN1C(=O)C(C)(C)c2cc(N)c(N)cc21

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 7/20 0.40
PTGS1 P23219 3/20 0.40
PTGS2 P35354 3/20 0.40
MGLL Q99685 2/20 0.40
FAAH O00519 1/20 0.40
CYP19A1 P11511 8/20 0.38
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6451576 0.95 MEN1 (0.39) SCN9APTGS1PTGS2MGLLFAAH
SCHEMBL2486662 0.89 PGR (0.37) CYP19A1
SCHEMBL13341347 0.85 ALDH1A1 (0.35)
SCHEMBL2486986 0.85 TDP1 (0.54) SCN9APTGS1PTGS2MGLLFAAH
SCHEMBL2491069 0.84 SCN9A (0.37) SCN9APTGS1PTGS2MGLLFAAH
SCHEMBL13341348 0.83 MPI (0.32)
SCHEMBL2486094 0.83 AURKA (0.44) MGLLCYP19A1
SCHEMBL2489388 0.82 ALDH1A1 (0.37)
SCHEMBL13341332 0.82 SCN9A (0.39) SCN9A
Hydrochloric Acid SCHEMBL10696532 0.81 AURKA (0.43) MGLLCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7714010-B2 Pyrrolobenzimidazolones and their use as anti-proliferative agents BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-05-11 US disclosed
US-7714010-B2 Pyrrolobenzimidazolones and their use as anti-proliferative agents BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-05-11 US disclosed
EP-1598353-A1 Pyrrolobenzimidazolones and their use as antiproliferative agents Boehringer Ingelheim International GmbH (DE) 2005-11-23 EP disclosed