SCHEMBL6451379

SCHEMBL6451379

Cn1c(=O)n(Cc2ccncc2)c(=O)c2cc(C(=O)OCc3ccccc3)sc21.O=C(OCc1ccccc1)c1cc2cncnc2s1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 5/20 0.43
HIF1A Q16665 2/20 0.40
MMP13 P45452 1/20 0.40
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CNR2 P34972 1/20 0.36
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6472710 0.89 TRPA1 (0.49) TRPA1HIF1AMMP13ALDH1A1MEN1
SCHEMBL6256050 0.89 TRPA1 (0.49) TRPA1HIF1AMMP13ALDH1A1MEN1
SCHEMBL6252686 0.84 MMP13 (0.53) TRPA1MMP13ALDH1A1MEN1KMT2A
SCHEMBL6916168 0.84 TRPA1 (0.42) TRPA1HIF1AMMP13ALDH1A1MEN1
SCHEMBL6255943 0.83 HIF1A (0.48) TRPA1HIF1AMMP13ALDH1A1HTT
SCHEMBL6445993 0.83 HIF1A (0.53) TRPA1HIF1AMMP13ALDH1A1HTT
SCHEMBL6254718 0.81 MMP13 (0.45) TRPA1HIF1AMMP13ALDH1A1MEN1
SCHEMBL6725010 0.81 TRPA1 (0.47) TRPA1HIF1AMMP13MEN1KMT2A
SCHEMBL6533924 0.81 MMP13 (0.49) TRPA1MMP13ALDH1A1MEN1KMT2A
SCHEMBL6730796 0.81 MMP13 (0.49) TRPA1MMP13ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1536786-A1 COMBINATION OF AN ALLOSTERIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2005-06-08 EP disclosed
WO-2004006913-A1 COMBINATION OF AN ALLOSTERIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed